Microwave-assisted simple synthesis of quinolines from anilines and alkyl vinyl ketones on the surface of silica gel in the presence of indium(III) chloride

被引：159

作者：

Ranu, BC ^{[1
]}

Hajra, A ^{[1
]}

Jana, U ^{[1
]}

机构：

[1] Indian Assoc Cultivat Sci, Dept Organ Chem, Calcutta 700032, W Bengal, India

来源：

TETRAHEDRON LETTERS | 2000年 / 41卷 / 04期

关键词：

quinolines; indium(III); chloride; microwave heating; silica gel;

D O I：

10.1016/S0040-4039(99)02111-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A simple and efficient procedure has been developed for the synthesis of 4-alkylquinolines by a one-pot reaction of anilines with alkyl vinyl ketones on the surface of silica gel impregnated with indium(III) chloride under microwave irradiation without any solvent. (C) 2000 Elsevier Science Ltd. All rights reserved.

引用

页码：531 / 533

页数：3

共 16 条

[1] Alhaider A. A., 1985, J MED CHEM, V28, P1398
[2] 2,4-DIAMINO-6,7-DIMETHOXYQUINOLINE DERIVATIVES AS ALPHA-1-ADRENOCEPTOR ANTAGONISTS AND ANTIHYPERTENSIVE AGENTS
CAMPBELL, SF
HARDSTONE, JD
PALMER, MJ
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (05) : 1031 - 1035
[3] Ruthenium-catalyzed synthesis of 2-ethyl-3-methylquinolines from anilines and triallylamine
Cho, CS
Oh, BH
Shim, SC
[J]. TETRAHEDRON LETTERS, 1999, 40 (08) : 1499 - 1500
[4] METHODOLOGIES FOR SYNTHESIS OF HETEROCYCLIC-COMPOUNDS
ISOBE, M
NISHIKAWA, T
YAMAMOTO, N
TSUKIYAMA, T
INO, A
OKITA, T
[J]. JOURNAL OF HETEROCYCLIC CHEMISTRY, 1992, 29 (03) : 619 - 625
[5] SYNTHESIS OF NITROGEN-HETEROCYCLES VIA PALLADIUM-CATALYZED INTRAMOLECULAR CYCLIZATION
LAROCK, RC
BABU, S
[J]. TETRAHEDRON LETTERS, 1987, 28 (44) : 5291 - 5294
[6] PALLADIUM-CATALYZED SYNTHESIS OF QUINOLINES FROM ALLYLIC ALCOHOLS AND ORTHO-IODOANILINE
LAROCK, RC
KUO, MY
[J]. TETRAHEDRON LETTERS, 1991, 32 (05) : 569 - 572
[7] Loh TP, 1998, SYNLETT, P975
[8] MANSKE RHF, 1953, ORG REACTIONS, V7, P59
[9] ANTIPROTOZOAL 4-ARYLOXY-2-AMINOQUINOLINES AND RELATED COMPOUNDS
MARKEES, DG
DEWEY, VC
KIDDER, GW
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1970, 13 (02) : 324 - &
[10] Quinoline, quinazoline and acridone alkaloids
Michael, JP
[J]. NATURAL PRODUCT REPORTS, 1997, 14 (06) : 605 - 618

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