Synthesis of Benzazoles by Hydrogen-Transfer Catalysis

被引：270

作者：

Blacker, A. John ^{[1
,2
]}

Farah, Mohamed M. ^{[1
,2
]}

Hall, Michael I. ^{[3
]}

Marsden, Stephen P. ^{[1
,2
]}

Saidi, Ourida ^{[3
]}

Williams, Jonathan M. J. ^{[3
]}

机构：

[1] Univ Leeds, Sch Chem, Leeds LS2 9JT, W Yorkshire, England

[2] Univ Leeds, Inst Proc Res & Dev, Leeds LS2 9JT, W Yorkshire, England

[3] Univ Bath, Dept Chem, Bath BA2 7AY, Avon, England

来源：

ORGANIC LETTERS | 2009年 / 11卷 / 09期

基金：

英国工程与自然科学研究理事会;

关键词：

ASYMMETRIC TRANSFER HYDROGENATION; ALCOHOLS; AMINES; OXIDATION; INHIBITORS; BENZIMIDAZOLES; LIGANDS; ESTERS; POTENT; AMIDES;

D O I：

10.1021/ol900557u

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Transition-metal-catalyzed hydrogen-transfer reactions have been used for the conversion of alcohols into benzimidazoles and aldehydes into benzoxazoles and benzothiazoles.

引用

页码：2039 / 2042

页数：4

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