Discovery of novel nonsteroidal glucocorticoid receptor modulators

被引：15

作者：

Link, JT

Sorensen, BK

Patel, J

Emery, M

Grynfarb, M

Goos-Nilsson, A

机构：

[1] Abbott Labs, Novum, Metab Dis Res, Dept 4CB, Abbott Pk, IL 60064 USA

[2] Abbott Labs, Medicinal Chem Technol, Abbott Pk, IL 60064 USA

[3] Karo Bio AB, SE-14157 Huddinge, Sweden

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 2004年 / 14卷 / 09期

关键词：

D O I：

10.1016/j.bmcl.2004.02.013

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

A new class of selective nonsteroidal glucocorticoid receptor modulators typified by N-{3-[benzyl-(4-chloro-2-fluorobenzyl)-amino]-2-methyl-phenyl -methanesulfonamide 19 has been discovered. (C) 2004 Elsevier Ltd. All rights reserved.

引用

页码：2209 / 2212

页数：4

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