Overview of the 2014 Food and Drug Administration Cardiovascular and Renal Drugs Advisory Committee Meeting About Vorapaxar

被引:37
作者
Baker, Nevin C. [1 ]
Lipinski, Michael J. [1 ]
Lhermusier, Thibault [1 ]
Waksman, Ron [1 ]
机构
[1] MedStar Washington Hosp Ctr, Dept Intervent Cardiol, Washington, DC 20010 USA
关键词
acute coronary syndrome; platelet aggregation inhibitors; thrombolytic therapy; PERCUTANEOUS CORONARY INTERVENTION; ACTIVATED RECEPTOR-1 ANTAGONIST; MYOCARDIAL-INFARCTION; SECONDARY PREVENTION; STROKE; DISCOVERY; THERAPY; DISEASE; UPDATE; TRENDS;
D O I
10.1161/CIRCULATIONAHA.114.011471
中图分类号
R5 [内科学];
学科分类号
100201 [内科学];
摘要
[No abstract available]
引用
收藏
页码:1287 / 1294
页数:8
相关论文
共 26 条
[1]
[Anonymous], PHARM THER S1
[2]
[Anonymous], EUR HEART J
[3]
[Anonymous], VOR NDA 204886 BRIEF
[4]
[Anonymous], US FOOD DRUG ADM PRE
[5]
[Anonymous], CLIN PHARM THER
[6]
Discovery of potent orally active thrombin receptor (protease activated receptor 1) antagonists as novel antithrombotic agents [J].
Chackalamannil, S ;
Xia, Y ;
Greenlee, WJ ;
Clasby, M ;
Doller, D ;
Tsai, H ;
Asberom, T ;
Czarniecki, M ;
Ahn, HS ;
Boykow, G ;
Foster, C ;
Agans-Fantuzzi, J ;
Bryant, M ;
Lau, J ;
Chintala, M .
JOURNAL OF MEDICINAL CHEMISTRY, 2005, 48 (19) :5884-5887
[7]
Discovery of a novel, orally active himbacine-based thrombin receptor antagonist (SCH 530348) with potent antiplatelet activity [J].
Chackalamannil, Samuel ;
Wang, Yuguang ;
Greenlee, William J. ;
Hu, Zhiyong ;
Xia, Yan ;
Ahn, Ho-Sam ;
Boykow, George ;
Hsieh, Yunsheng ;
Palamanda, Jairam ;
Agans-Fantuzzi, Jacqueline ;
Kurowski, Stan ;
Graziano, Michael ;
Chintala, Madhu .
JOURNAL OF MEDICINAL CHEMISTRY, 2008, 51 (11) :3061-3064
[8]
Thrombin receptor (protease activated receptor-1) antagonists as potent antithrombotic agents with strong antiplatelet effects [J].
Chackalamannil, Samuel .
JOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (18) :5389-5403
[9]
SCH 602539, a Protease-Activated Receptor-1 Antagonist, Inhibits Thrombosis Alone and in Combination With Cangrelor in a Folts Model of Arterial Thrombosis in Cynomolgus Monkeys [J].
Chintala, Madhu ;
Strony, John ;
Yang, Bo ;
Kurowski, Stan ;
Li, Qiu .
ARTERIOSCLEROSIS THROMBOSIS AND VASCULAR BIOLOGY, 2010, 30 (11) :2143-2149
[10]
Collins R, 2009, LANCET, V373, P1849, DOI 10.1016/S0140-6736(09)60503-1