Synthesis and reactivity of alkyl (4-aminothien-3-yl)carbamates

被引：6

作者：

Brugier, D ^{[1
]}

Outurquin, F ^{[1
]}

Paulmier, C ^{[1
]}

机构：

[1] UNIV ROUEN,UFR SCI & TECH,IRCOF,SYNTHESE THIO & SELENOORGAN LAB,F-76821 MONT ST AIGNAN,FRANCE

来源：

TETRAHEDRON | 1997年 / 53卷 / 30期

关键词：

D O I：

10.1016/S0040-4020(97)00681-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Monocarbomates 2 have been prepared from 3,4-diaminothiophene 1 and were alkylated on the thiophene nucleus using an aldehyde and selenophenol, under acid catalysis. This reaction has allowed the access to 2-alkyl 3,4-diaminothiophenes 9,3,5-diaminodithieno[3,2-b:2',3'-e]pyridines 10 and 1-alkyl thieno[3,4-d]imidazolones 13. (C) 1997 Elsevier Science Ltd.

引用

页码：10331 / 10344

页数：14

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