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Drug delivery systems .2. Camptothecin 20-O-poly(ethylene glycol)ester transport forms
被引:95
作者
:
Greenwald, RB
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Greenwald, RB
Pendri, A
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Pendri, A
Conover, C
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Conover, C
Gilbert, C
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Gilbert, C
Yang, R
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Yang, R
Xia, J
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Xia, J
机构
:
[1]
Enzon Inc., Piscataway, NJ 08854-3969
来源
:
JOURNAL OF MEDICINAL CHEMISTRY
|
1996年
/ 39卷
/ 10期
关键词
:
D O I
:
10.1021/jm9600555
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
[No abstract available]
引用
收藏
页码:1938 / 1940
页数:3
相关论文
共 13 条
[1]
BUNDGAARD H, 1986, BIOREVERSIBLE DERIVA, P49
[2]
THE STRUCTURAL BASIS OF CAMPTOTHECIN INTERACTIONS WITH HUMAN SERUM-ALBUMIN - IMPACT ON DRUG STABILITY
BURKE, TG
论文数:
0
引用数:
0
h-index:
0
机构:
OHIO STATE UNIV,COLL PHARM,DIV PHARMACEUT,COLUMBUS,OH 43210
BURKE, TG
MI, ZH
论文数:
0
引用数:
0
h-index:
0
机构:
OHIO STATE UNIV,COLL PHARM,DIV PHARMACEUT,COLUMBUS,OH 43210
MI, ZH
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1994,
37
(01)
: 40
-
46
[3]
Garzon-Aburbeh A., 1990, [No title captured], Patent No. 4943579
[4]
Drug delivery systems: Water soluble taxol 2'-poly(ethylene glycol) ester prodrugs - Design and in vivo effectiveness
Greenwald, RB
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Greenwald, RB
Gilbert, CW
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Gilbert, CW
Pendri, A
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Pendri, A
Conover, CD
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Conover, CD
Xia, J
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Xia, J
Martinez, A
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Martinez, A
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1996,
39
(02)
: 424
-
431
[5]
MODIFICATION OF THE HYDROXY LACTONE RING OF CAMPTOTHECIN - INHIBITION OF MAMMALIAN TOPOISOMERASE-I AND BIOLOGICAL-ACTIVITY
HERTZBERG, RP
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
HERTZBERG, RP
CARANFA, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
CARANFA, MJ
HOLDEN, KG
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
HOLDEN, KG
JAKAS, DR
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
JAKAS, DR
GALLAGHER, G
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
GALLAGHER, G
MATTERN, MR
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
MATTERN, MR
MONG, SM
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
MONG, SM
BARTUS, JO
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
BARTUS, JO
JOHNSON, RK
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
JOHNSON, RK
KINGSBURY, WD
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
KINGSBURY, WD
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1989,
32
(03)
: 715
-
720
[6]
JAXEL C, 1989, CANCER RES, V49, P1465
[7]
SYNTHESIS AND ANTITUMOR-ACTIVITY OF NOVEL WATER-SOLUBLE DERIVATIVES OF CAMPTOTHECIN AS SPECIFIC INHIBITORS OF TOPOISOMERASE-I
LUZZIO, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
LUZZIO, MJ
BESTERMAN, JM
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
BESTERMAN, JM
EMERSON, DL
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
EMERSON, DL
EVANS, MG
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
EVANS, MG
LACKEY, K
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
LACKEY, K
LEITNER, PL
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
LEITNER, PL
MCINTYRE, G
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
MCINTYRE, G
MORTON, B
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
MORTON, B
MYERS, PL
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
MYERS, PL
PEEL, M
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
PEEL, M
SISCO, JM
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
SISCO, JM
STERNBACH, DD
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
STERNBACH, DD
TONG, WQ
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
TONG, WQ
TRUESDALE, A
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
TRUESDALE, A
UEHLING, DE
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
UEHLING, DE
VUONG, A
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
VUONG, A
YATES, J
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
YATES, J
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1995,
38
(03)
: 395
-
401
[8]
DIFFERENTIAL INTERACTIONS OF CAMPTOTHECIN LACTONE AND CARBOXYLATE FORMS WITH HUMAN BLOOD COMPONENTS
MI, ZH
论文数:
0
引用数:
0
h-index:
0
机构:
OHIO STATE UNIV, COLL PHARM, DIV PHARMACEUT, COLUMBUS, OH 43210 USA
MI, ZH
BURKE, TG
论文数:
0
引用数:
0
h-index:
0
机构:
OHIO STATE UNIV, COLL PHARM, DIV PHARMACEUT, COLUMBUS, OH 43210 USA
BURKE, TG
[J].
BIOCHEMISTRY,
1994,
33
(34)
: 10325
-
10336
[9]
MARKED INTERSPECIES VARIATIONS CONCERNING THE INTERACTIONS OF CAMPTOTHECIN WITH SERUM ALBUMINS - A FREQUENCY-DOMAIN FLUORESCENCE SPECTROSCOPIC STUDY
MI, ZH
论文数:
0
引用数:
0
h-index:
0
机构:
OHIO STATE UNIV,COLL PHARM,DIV PHARMACEUT,COLUMBUS,OH 43210
MI, ZH
BURKE, TG
论文数:
0
引用数:
0
h-index:
0
机构:
OHIO STATE UNIV,COLL PHARM,DIV PHARMACEUT,COLUMBUS,OH 43210
BURKE, TG
[J].
BIOCHEMISTRY,
1994,
33
(42)
: 12540
-
12545
[10]
POTMESIL M, 1994, CANCER RES, V54, P1431
←
1
2
→
共 13 条
[1]
BUNDGAARD H, 1986, BIOREVERSIBLE DERIVA, P49
[2]
THE STRUCTURAL BASIS OF CAMPTOTHECIN INTERACTIONS WITH HUMAN SERUM-ALBUMIN - IMPACT ON DRUG STABILITY
BURKE, TG
论文数:
0
引用数:
0
h-index:
0
机构:
OHIO STATE UNIV,COLL PHARM,DIV PHARMACEUT,COLUMBUS,OH 43210
BURKE, TG
MI, ZH
论文数:
0
引用数:
0
h-index:
0
机构:
OHIO STATE UNIV,COLL PHARM,DIV PHARMACEUT,COLUMBUS,OH 43210
MI, ZH
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1994,
37
(01)
: 40
-
46
[3]
Garzon-Aburbeh A., 1990, [No title captured], Patent No. 4943579
[4]
Drug delivery systems: Water soluble taxol 2'-poly(ethylene glycol) ester prodrugs - Design and in vivo effectiveness
Greenwald, RB
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Greenwald, RB
Gilbert, CW
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Gilbert, CW
Pendri, A
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Pendri, A
Conover, CD
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Conover, CD
Xia, J
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Xia, J
Martinez, A
论文数:
0
引用数:
0
h-index:
0
机构:
Enzon Inc., Piscataway, NJ 08854-3969
Martinez, A
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1996,
39
(02)
: 424
-
431
[5]
MODIFICATION OF THE HYDROXY LACTONE RING OF CAMPTOTHECIN - INHIBITION OF MAMMALIAN TOPOISOMERASE-I AND BIOLOGICAL-ACTIVITY
HERTZBERG, RP
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
HERTZBERG, RP
CARANFA, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
CARANFA, MJ
HOLDEN, KG
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
HOLDEN, KG
JAKAS, DR
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
JAKAS, DR
GALLAGHER, G
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
GALLAGHER, G
MATTERN, MR
论文数:
0
引用数:
0
h-index:
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机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
MATTERN, MR
MONG, SM
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
MONG, SM
BARTUS, JO
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
BARTUS, JO
JOHNSON, RK
论文数:
0
引用数:
0
h-index:
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机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
JOHNSON, RK
KINGSBURY, WD
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DEPT MOLEC PHARMACOL,KING OF PRUSSIA,PA 19406
KINGSBURY, WD
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1989,
32
(03)
: 715
-
720
[6]
JAXEL C, 1989, CANCER RES, V49, P1465
[7]
SYNTHESIS AND ANTITUMOR-ACTIVITY OF NOVEL WATER-SOLUBLE DERIVATIVES OF CAMPTOTHECIN AS SPECIFIC INHIBITORS OF TOPOISOMERASE-I
LUZZIO, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
LUZZIO, MJ
BESTERMAN, JM
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
BESTERMAN, JM
EMERSON, DL
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
EMERSON, DL
EVANS, MG
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
EVANS, MG
LACKEY, K
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
LACKEY, K
LEITNER, PL
论文数:
0
引用数:
0
h-index:
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机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
LEITNER, PL
MCINTYRE, G
论文数:
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引用数:
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h-index:
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GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
MCINTYRE, G
MORTON, B
论文数:
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引用数:
0
h-index:
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机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
MORTON, B
MYERS, PL
论文数:
0
引用数:
0
h-index:
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机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
MYERS, PL
PEEL, M
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
PEEL, M
SISCO, JM
论文数:
0
引用数:
0
h-index:
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机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
SISCO, JM
STERNBACH, DD
论文数:
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引用数:
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h-index:
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GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
STERNBACH, DD
TONG, WQ
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引用数:
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h-index:
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GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
TONG, WQ
TRUESDALE, A
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引用数:
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GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
TRUESDALE, A
UEHLING, DE
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引用数:
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h-index:
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GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
UEHLING, DE
VUONG, A
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VUONG, A
YATES, J
论文数:
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引用数:
0
h-index:
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机构:
GLAXO INC,RES INST,DEPT CELL BIOL,RES TRIANGLE PK,NC 27709
YATES, J
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1995,
38
(03)
: 395
-
401
[8]
DIFFERENTIAL INTERACTIONS OF CAMPTOTHECIN LACTONE AND CARBOXYLATE FORMS WITH HUMAN BLOOD COMPONENTS
MI, ZH
论文数:
0
引用数:
0
h-index:
0
机构:
OHIO STATE UNIV, COLL PHARM, DIV PHARMACEUT, COLUMBUS, OH 43210 USA
MI, ZH
BURKE, TG
论文数:
0
引用数:
0
h-index:
0
机构:
OHIO STATE UNIV, COLL PHARM, DIV PHARMACEUT, COLUMBUS, OH 43210 USA
BURKE, TG
[J].
BIOCHEMISTRY,
1994,
33
(34)
: 10325
-
10336
[9]
MARKED INTERSPECIES VARIATIONS CONCERNING THE INTERACTIONS OF CAMPTOTHECIN WITH SERUM ALBUMINS - A FREQUENCY-DOMAIN FLUORESCENCE SPECTROSCOPIC STUDY
MI, ZH
论文数:
0
引用数:
0
h-index:
0
机构:
OHIO STATE UNIV,COLL PHARM,DIV PHARMACEUT,COLUMBUS,OH 43210
MI, ZH
BURKE, TG
论文数:
0
引用数:
0
h-index:
0
机构:
OHIO STATE UNIV,COLL PHARM,DIV PHARMACEUT,COLUMBUS,OH 43210
BURKE, TG
[J].
BIOCHEMISTRY,
1994,
33
(42)
: 12540
-
12545
[10]
POTMESIL M, 1994, CANCER RES, V54, P1431
←
1
2
→