An improved synthesis of the anti-picornavirus flavone 3-O-methylquercetin

被引：9

作者：

Boers, F ^{[1
]}

Deng, BL ^{[1
]}

Lemiere, G ^{[1
]}

Lepoivre, J ^{[1
]}

DeGroot, A ^{[1
]}

Dommisse, R ^{[1
]}

Vlietinck, AJ ^{[1
]}

机构：

[1] UNIV ANTWERP,UIA,DEPT PHARMACEUT SCI,B-2610 ANTWERP,BELGIUM

来源：

ARCHIV DER PHARMAZIE | 1997年 / 330卷 / 9-10期

关键词：

3-O-methylquercetin; anti-picornavirus flavones; Allan-Robinson condensation; Baker-Venkataraman transformation; phase transfer catalysis;

D O I：

10.1002/ardp.19973300909

中图分类号：

R914 [药物化学];

学科分类号：

100701 [药物化学];

摘要：

Two optimised procedures to synthesise 3-O-methylquercetin (1), an important antivirally active flavone, are presented: one is based on an Allan-Robinson condensation, the other one on a modified phase transfer catalysed Baker-Venkataraman transformation.

引用

页码：313 / 316

页数：4

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