A facile method for the transformation of N-(tert-butoxycarbonyl) α-amino acids to N-unprotected α-amino methyl esters

被引：25

作者：

Chen, BC ^{[1
]}

Skoumbourdis, AP ^{[1
]}

Guo, P ^{[1
]}

Bednarz, MS ^{[1
]}

Kocy, OR ^{[1
]}

Sundeen, JE ^{[1
]}

Vite, GD ^{[1
]}

机构：

[1] Bristol Myers Squibb Pharmaceut Res Inst, Princeton, NJ 08543 USA

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1999年 / 64卷 / 25期

关键词：

D O I：

10.1021/jo990311w

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[No abstract available]

引用

页码：9294 / 9296

页数：3

共 48 条

[1] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF KETOMETHYLENE-CONTAINING NONAPEPTIDE ANALOGS OF SNAKE-VENOM ANGIOTENSIN CONVERTING ENZYME-INHIBITORS [J].

ALMQUIST, RG ;

CHAO, WR ;

JUDD, AK ;

MITOMA, C ;

ROSSI, DJ ;

PANASEVICH, RE ;

MATTHEWS, RJ .

JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (03) :561-567

[2] Diastereoselective palladium(0)-catalyzed azidation of 1-alkenylcyclopropyl esters:: asymmetric synthesis of (-)-(1R,2S)-norcoronamic acid [J].

Atlan, V ;

Racouchot, S ;

Rubin, M ;

Bremer, C ;

Ollivier, J ;

de Meijere, A ;

Salaün, J .

TETRAHEDRON-ASYMMETRY, 1998, 9 (07) :1131-1135

[3]

Badorrey R, 1997, SYNTHESIS-STUTTGART, P747

[4] SYNTHESIS OF 4-PHOSPHONO-DL-PHENYLALANINE AND OF 4-(PHOSPHONOMETHYL)-DL-PHENYLALANINE, 2 ANALOGS OF O-PHOSPHOTYROSINE [J].

BAYLELACOSTE, M ;

MOULINES, J ;

COLLIGNON, N ;

BOUMEKOUEZ, A ;

DETINGUYMOREAUD, E ;

NEUZIL, E .

TETRAHEDRON, 1990, 46 (23) :7793-7802

[5]

BELAGALI SL, 1995, INDIAN J CHEM B, V34, P45

[6] STUDIES ON THE TOTAL SYNTHESIS OF BOUVARDIN AND DEOXYBOUVARDIN - CYCLIC HEXAPEPTIDE CYCLIZATION STUDIES AND PREPARATION OF KEY PARTIAL STRUCTURES [J].

BOGER, DL ;

YOHANNES, D .

JOURNAL OF ORGANIC CHEMISTRY, 1988, 53 (03) :487-499

[7] RENIN INHIBITORS - SYNTHESES OF SUBNANOMOLAR, COMPETITIVE, TRANSITION-STATE ANALOG INHIBITORS CONTAINING A NOVEL ANALOG OF STATINE [J].

BOGER, J ;

PAYNE, LS ;

PERLOW, DS ;

LOHR, NS ;

POE, M ;

BLAINE, EH ;

ULM, EH ;

SCHORN, TW ;

LAMONT, BI ;

LIN, TY ;

KAWAI, M ;

RICH, DH ;

VEBER, DF .

JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (12) :1779-1790

[8] Synthesis of modified carboxyl binding pockets of vancomycin and teicoplanin [J].

BoisChoussy, M ;

Neuville, L ;

Beugelmans, R ;

Zhu, JP .

JOURNAL OF ORGANIC CHEMISTRY, 1996, 61 (26) :9309-9322

[9] TOTAL SYNTHESIS OF 6-DEOXY-6-AMINOHEPTOPYRANURONIC ACID-DERIVATIVES [J].

CASIRAGHI, G ;

COLOMBO, L ;

RASSU, G ;

SPANU, P .

JOURNAL OF ORGANIC CHEMISTRY, 1991, 56 (23) :6523-6527

[10] ENANTIOSELECTIVE SYNTHESIS OF PRIMARY AMINES VIA GRIGNARD ADDITIONS TO STEREOGENIC N-(ALPHA-PHENYL-BETA-(BENZYLOXY)ETHYL)NITRONES [J].

CHANG, ZY ;

COATES, RM .

JOURNAL OF ORGANIC CHEMISTRY, 1990, 55 (11) :3475-3483

← 1 2 3 4 5 →