Total synthesis of (-)-epothilone B: An extension of the Suzuki coupling method and insights into structure-activity relationships of the epothilones

被引:152
作者
Su, DS
Meng, DF
Bertinato, P
Balog, A
Sorensen, EJ
Danishefsky, SJ
Zheng, YH
Chou, TC
He, LF
Horwitz, SB
机构
[1] SLOAN KETTERING INST CANC RES,BIOORGAN CHEM LAB,NEW YORK,NY 10021
[2] SLOAN KETTERING INST,BIOCHEM PHARMACOL LAB,NEW YORK,NY
[3] YESHIVA UNIV ALBERT EINSTEIN COLL MED,DEPT MOL PHARMACOL,BRONX,NY 10461
[4] COLUMBIA UNIV,DEPT CHEM,NEW YORK,NY 10027
来源
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH | 1997年 / 36卷 / 07期
关键词
antitumor agents; epothilone; natural products; total synthesis;
D O I
10.1002/anie.199707571
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
[No abstract available]
引用
收藏
页码:757 / 759
页数:3
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