Three component synthesis of β-amino carbonyl compounds using indium trichloride-catalyzed one-pot Mannich-type reaction in water

被引：167

作者：

Loh, TP ^{[1
]}

Liung, SBKW ^{[1
]}

Tan, KL ^{[1
]}

Wei, LL ^{[1
]}

机构：

[1] Natl Univ Singapore, Dept Chem, Singapore 119260, Singapore

来源：

TETRAHEDRON | 2000年 / 56卷 / 20期

关键词：

D O I：

10.1016/S0040-4020(00)00221-0

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The use of indium trichloride as catalyst in a one-pot Mannich reaction in water gives high yields for the formation of beta-aminoketones/esters/acids is described. The catalyst can be recycled when the reaction is complete (Loh T.-P.; Wei L.-L. Tetrahedron Lett. 1998, 39, 323). (C) 2000 Elsevier Science Ltd. All rights reserved.

引用

页码：3227 / 3237

页数：11

共 34 条

[1] Akiyama T, 1999, SYNLETT, P1426
[2] HBF4 catalyzed Mannich-type reaction in aqueous media
Akiyama, T
Takaya, J
Kagoshima, H
[J]. SYNLETT, 1999, (07) : 1045 - 1048
[3] [Anonymous], [No title captured]
[4] Arend M, 1998, ANGEW CHEM INT EDIT, V37, P1044, DOI 10.1002/(SICI)1521-3773(19980504)37:8<1044::AID-ANIE1044>3.0.CO
[5] 2-E
[6] A NEW SYNTHESIS OF 1-TERT-BUTYLDIMETHYLSILYL-3-ACETYL-4-CARBOXYAZETIDIN-2-ONE
CAINELLI, G
CONTENTO, M
DRUSIANI, A
PANUNZIO, M
PLESSI, L
[J]. JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1985, (04) : 240 - 240
[7] Highly diastereoselective addition of silyl enolates to chiral imines derived from (S)-valine methyl ester using lanthanide triflate.
Cozzi, PG
DiSimone, B
UmaniRonchi, A
[J]. TETRAHEDRON LETTERS, 1996, 37 (10) : 1691 - 1694
[8] SYNTHETIC STUDIES TOWARD AFLAVININE - A SYNTHESIS OF 3-DESMETHYLAFLAVININE VIA A [2 + 2 + 2] ANNULATION
DANISHEFSKY, S
CHACKALAMANNIL, S
HARRISON, P
SILVESTRI, M
COLE, P
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1985, 107 (08) : 2474 - 2484
[9] KETENE BIS(TRIMETHYLSILYL) ACETALS - CROSS-ALDOL TYPE CONDENSATION-REACTIONS WITH ALDEHYDES AND SCHIFF-BASES
DUBOIS, JE
AXIOTIS, G
[J]. TETRAHEDRON LETTERS, 1984, 25 (20) : 2143 - 2146
[10] Evans D. A., 1982, TOP STEREOCHEM, V13, P1, DOI DOI 10.1002/9780470147221.CHL

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