The Friedlander synthesis of 4-perfluoroalkylquinolines

被引：99

作者：

Strekowski, L ^{[1
]}

Czarny, A ^{[1
]}

Lee, H ^{[1
]}

机构：

[1] Georgia State Univ, Dept Chem, Atlanta, GA 30303 USA

来源：

JOURNAL OF FLUORINE CHEMISTRY | 2000年 / 104卷 / 02期

关键词：

2-perfluoroacylanilines; ketones; beta-diketones; benzoylacetonitrile; condensation;

D O I：

10.1016/S0022-1139(00)00252-9

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

2-Substituted and 2,3-disubstituted 4-perfluoroalkylquinolines are obtained in high yield by the acid-catalyzed reaction of 2-perfluoroacylanilines with enolizable ketones and beta-diketones. (C) 2000 Elsevier Science S.A. All rights reserved.

引用

页码：281 / 284

页数：4

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