A novel approach for the synthesis of 5-substituted tetrazole derivatives from primary amides in mild one-step method.

被引：45

作者：

ElAhl, AAS ^{[1
]}

Elmorsy, SS ^{[1
]}

Elbeheery, AH ^{[1
]}

Amer, FA ^{[1
]}

机构：

[1] MANSOURA UNIV,FAC SCI,DEPT CHEM,MANSOURA,EGYPT

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 07期

关键词：

D O I：

10.1016/S0040-4039(97)00052-X

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A new mild one-step method for the conversion of primary acid amides to 5-substituted tetrazoles in nearly quantitative yields employing triazidochlorosilane (TACS) is reported. (C) 1997, Elsevier Science Ltd.

引用

页码：1257 / 1260

页数：4

共 16 条

[1] TETRAZOLYL PEPTIDES AND THE TETRAZOLE ANALOG OF 3-AMINONOCARDICINIC ACID [J].

ANDERSON, DW ;

CAMPBELL, MM ;

MALIK, M .

TETRAHEDRON LETTERS, 1990, 31 (12) :1755-1758

[2] A STUDY OF THE STRUCTURE OF SOME CYCLIC AMIDES AND RELATED TETRAZOLES [J].

BURKE, RL ;

HERBST, RM .

JOURNAL OF ORGANIC CHEMISTRY, 1955, 20 (06) :726-735

[3]

BUTLER RN, 1984, COMPREHENSIVE HETERO, V5, P791

[4] 3 SYNTHETIC ROUTES TO A STERICALLY HINDERED TETRAZOLE - A NEW ONE-STEP MILD CONVERSION OF AN AMIDE INTO A TETRAZOLE [J].

DUNCIA, JV ;

PIERCE, ME ;

SANTELLA, JB .

JOURNAL OF ORGANIC CHEMISTRY, 1991, 56 (07) :2395-2400

[5]

Eiichi Kano, Patent No. [60, 130, 572, 60130572]

[6] A FACILE AND CONVENIENT SYNTHESIS OF SUBSTITUTED TETRAZOLE DERIVATIVES FROM KETONES OR ALPHA-BETA-UNSATURATED KETONES [J].

ELAHL, AAS ;

ELMORSY, SS ;

SOLIMAN, H ;

AMER, FA .

TETRAHEDRON LETTERS, 1995, 36 (40) :7337-7340

[7] OXIDATION OF ALDEHYDES TO ACYL AZIDES USING TRIAZIDOCHLOROSILANE (TACS)-ACTIVE MANGANESE-DIOXIDE REAGENT [J].

ELMORSY, SS .

TETRAHEDRON LETTERS, 1995, 36 (08) :1341-1342

[8] SYNTHESIS OF TRIAZIDOCHLOROSILANE (TACS) - A NOVEL SILICON MEDIATED ONE-POT CONVERSION OF ALDEHYDES TO NITRILES [J].

ELMORSY, SS ;

EIAHL, AAS ;

SOLIMAN, H ;

AMER, FA .

TETRAHEDRON LETTERS, 1995, 36 (15) :2639-2640

[9] SYNTHESIS OF 1-SUBSTITUTED TETRAZOLES [J].

FALLON, FG ;

HERBST, RM .

JOURNAL OF ORGANIC CHEMISTRY, 1957, 22 (08) :933-936

[10] APPARENT ACIDIC DISSOCIATION OF SOME 5-ARYLTETRAZOLES [J].

HERBST, RM ;

WILSON, KR .

JOURNAL OF ORGANIC CHEMISTRY, 1957, 22 (10) :1142-1145

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