Selective cyclooxygenase-2 inhibitors

被引:89
作者
Prasit, P
Riendeau, D
机构
[1] Merck Frosst Centre for Therapeutic Research, Pointe Claire-Dorval, Que. H9R 4P8
来源
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 32 | 1997年 / 32卷
关键词
D O I
10.1016/S0065-7743(08)61479-7
中图分类号
O69 [应用化学];
学科分类号
081704 ;
摘要
[No abstract available]
引用
收藏
页码:211 / 220
页数:10
相关论文
共 81 条
  • [1] Adams J, 1996, J NEUROCHEM, V66, P6
  • [2] PURIFICATION, CHARACTERIZATION AND SELECTIVE-INHIBITION OF HUMAN PROSTAGLANDIN-G/H SYNTHASE-1 AND SYNTHASE-2 EXPRESSED IN THE BACULOVIRUS SYSTEM
    BARNETT, J
    CHOW, J
    IVES, D
    CHIOU, M
    MACKENZIE, R
    OSEN, E
    NGUYEN, B
    TSING, S
    BACH, C
    FREIRE, J
    CHAN, H
    SIGAL, E
    RAMESHA, C
    [J]. BIOCHIMICA ET BIOPHYSICA ACTA-PROTEIN STRUCTURE AND MOLECULAR ENZYMOLOGY, 1994, 1209 (01): : 130 - 139
  • [3] Barnett JW, Eur. Pat Appl., Patent No. [714895, EP 714895]
  • [4] BATT DG, Patent No. 9610012
  • [5] Bertenshaw S. R., [No title captured], Patent No. [WO 9515316, 9515316]
  • [6] BESWICK PJ, Patent No. 9631509
  • [7] BLACK C, Patent No. 9636623
  • [8] BLACK C, Patent No. 9619469
  • [9] From indomethacin to a selective COX-2 inhibitor: Development of indolalkanoic acids as potent and selective cyclooxygenase-2 inhibitors
    Black, WC
    Bayly, C
    Belley, M
    Chan, CC
    Charleson, S
    Denis, D
    Gauthier, JY
    Gordon, R
    Guay, D
    Kargman, S
    Lau, CK
    Leblanc, Y
    Mancini, J
    Ouellet, M
    Percival, D
    Roy, P
    Skorey, K
    Tagari, P
    Vickers, P
    Wong, E
    Xu, L
    Prasit, P
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1996, 6 (06) : 725 - 730
  • [10] A human whole blood assay for clinical evaluation of biochemical efficacy of cyclooxygenase inhibitors
    Brideau, C
    Kargman, S
    Liu, S
    Dallob, AL
    Ehrich, EW
    Rodger, IW
    Chan, CC
    [J]. INFLAMMATION RESEARCH, 1996, 45 (02) : 68 - 74