Similarities and distinctions in the mode of action of different classes of antioestrogens

被引：156

作者：

Wakeling, AE ^{[1
]}

机构：

[1] AstraZeneca, Canc & Infect Biosci Dept, Macclesfield SK10 4TG, Cheshire, England

来源：

关键词：

D O I：

10.1677/erc.0.0070017

中图分类号：

R73 [肿瘤学];

学科分类号：

100214 ;

摘要：

[No abstract available]

引用

页码：17 / 28

页数：12

共 148 条

[1]

ALBERT JL, 1990, CANCER RES, V50, P3306

[2] STIMULATION OF ESTROGEN RECEPTOR-MEDIATED TRANSCRIPTION AND ALTERATION IN THE PHOSPHORYLATION STATE OF THE RAT UTERINE ESTROGEN-RECEPTOR BY ESTROGEN, CYCLIC ADENOSINE-MONOPHOSPHATE, AND INSULIN-LIKE GROWTH FACTOR-I [J].

ARONICA, SM ;

KATZENELLENBOGEN, BS .

MOLECULAR ENDOCRINOLOGY, 1993, 7 (06) :743-752

[3] Reproductive endocrine and endometrial effects of raloxifene hydrochloride, a selective estrogen receptor modulator, in women with regular menstrual cycles [J].

Baker, VL ;

Draper, M ;

Paul, S ;

Allerheiligen, S ;

Glant, M ;

Shifren, J ;

Jaffe, RB .

JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1998, 83 (01) :6-13

[4] GENE-REGULATION BY STEROID-HORMONES [J].

BEATO, M .

CELL, 1989, 56 (03) :335-344

[5] ROLE OF THE 2 ACTIVATING DOMAINS OF THE ESTROGEN-RECEPTOR IN THE CELL-TYPE AND PROMOTER-CONTEXT DEPENDENT AGONISTIC ACTIVITY OF THE ANTIESTROGEN 4-HYDROXYTAMOXIFEN [J].

BERRY, M ;

METZGER, D ;

CHAMBON, P .

EMBO JOURNAL, 1990, 9 (09) :2811-2818

[6] UTERINE BIOASSAY OF TAMOXIFEN, TRIOXIFENE AND A NEW ESTROGEN ANTAGONIST (LY117018) IN RATS AND MICE [J].

BLACK, LJ ;

GOODE, RL .

LIFE SCIENCES, 1980, 26 (17) :1453-1458

[7] CONTRASTING EFFECTS OF TAMOXIFEN AND ICI-182-780 ON ESTROGEN-INDUCED CALBINDIN-D9K GENE-EXPRESSION IN THE UTERUS AND IN PRIMARY CULTURE OF MYOMETRIAL CELLS [J].

BLIN, C ;

LHORSET, F ;

LECLERC, T ;

LAMBERT, M ;

COLNOT, S ;

THOMASSET, M ;

PERRET, C .

JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1995, 55 (01) :1-7

[8] Estrogenic and antiestrogenic regulation of the half-life of covalently labeled estrogen receptor in MCF-7 breast cancer cells [J].

Borras, M ;

Laios, I ;

ElKhissiin, A ;

Seo, HS ;

Lempereur, F ;

Legros, N ;

Leclercq, G .

JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1996, 57 (3-4) :203-213

[9]

BOWLER J, 1989, Steroids, V54, P71, DOI 10.1016/0039-128X(89)90076-7

[10] DROLOXIFENE, A NEW ANTIESTROGEN IN POSTMENOPAUSAL ADVANCED BREAST-CANCER - PRELIMINARY-RESULTS OF A DOUBLE-BLIND DOSE-FINDING PHASE-II TRIAL [J].

BRUNING, PF .

EUROPEAN JOURNAL OF CANCER, 1992, 28A (8-9) :1404-1407

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