Plasma protein binding of drugs

被引:347
作者
Olson, RE
Christ, DD
机构
[1] The DuPont Merck Pharmaceutical Company Wilmington
来源
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 31 | 1996年 / 31卷
关键词
D O I
10.1016/S0065-7743(08)60472-8
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:327 / 336
页数:10
相关论文
共 87 条
[1]   THERMODYNAMIC ASPECTS OF THE MOLECULAR RECOGNITION OF DRUGS BY HUMAN SERUM-ALBUMIN [J].
AKI, H ;
GOTO, M ;
YAMAMOTO, M .
THERMOCHIMICA ACTA, 1995, 251 :379-388
[2]   THERMODYNAMIC CHARACTERIZATION OF DRUG-BINDING TO HUMAN SERUM-ALBUMIN BY ISOTHERMAL TITRATION MICROCALORIMETRY [J].
AKI, H ;
YAMAMOTO, M .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1994, 83 (12) :1712-1716
[3]   MICRODIALYSIS SAMPLING TO DETERMINE THE PHARMACOKINETICS OF UNBOUND SDZ-ICM-567 IN BLOOD AND BRAIN IN AWAKE, FREELY-MOVING RATS [J].
ALONSO, MJ ;
BRUELISAUER, A ;
MISSLIN, P ;
LEMAIRE, M .
PHARMACEUTICAL RESEARCH, 1995, 12 (02) :291-294
[4]   STEREOSPECIFIC AND COMPETITIVE-BINDING OF DRUGS TO HUMAN SERUM-ALBUMIN - A DIFFERENCE CIRCULAR-DICHROISM APPROACH [J].
ASCOLI, G ;
BERTUCCI, C ;
SALVADORI, P .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1995, 84 (06) :737-741
[5]  
BEAUCHAMP HT, 1995, J PHARMACOL EXP THER, V272, P612
[6]  
BIELLO JA, 1995, ANTIMICROB AGENTS CH, V39, P2523
[7]   AN INVESTIGATION OF THE USE OF NILE-RED AS A LONG-WAVELENGTH FLUORESCENT-PROBE FOR THE STUDY OF ALPHA(1)-ACID GLYCOPROTEIN-DRUG INTERACTIONS [J].
BROWN, MB ;
MILLER, JN ;
SEARE, NJ .
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 1995, 13 (08) :1011-1017
[8]   SC-52151, A NOVEL INHIBITOR OF THE HUMAN-IMMUNODEFICIENCY-VIRUS PROTEASE [J].
BRYANT, M ;
GETMAN, D ;
SMIDT, M ;
MARR, J ;
CLARE, M ;
DILLARD, R ;
LANSKY, D ;
DECRESCENZO, G ;
HEINTZ, R ;
HOUSEMAN, K ;
REED, K ;
STOLZENBACH, J ;
TALLEY, J ;
VAZQUEZ, M ;
MUELLER, R .
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1995, 39 (10) :2229-2234
[9]  
CARTER DC, 1994, ADV PROTEIN CHEM, V45, P153
[10]   PRELIMINARY CRYSTALLOGRAPHIC STUDIES OF 4 CRYSTAL FORMS OF SERUM-ALBUMIN [J].
CARTER, DC ;
CHANG, B ;
HO, JX ;
KEELING, K ;
KRISHNASAMI, Z .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1994, 226 (03) :1049-1052