Syntheses and antifungal activity of pseudomycin side-chain analogues. Part 1

被引：12

作者：

Jamison, J ^{[1
]}

Levy, S ^{[1
]}

Sun, XC ^{[1
]}

Zeckner, D ^{[1
]}

Current, W ^{[1
]}

Zweifel, M ^{[1
]}

Rodriguez, M ^{[1
]}

Turner, W ^{[1
]}

Chen, SH ^{[1
]}

机构：

[1] Lilly Res Labs, Indianapolis, IN 46285 USA

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 2000年 / 10卷 / 18期

关键词：

D O I：

10.1016/S0960-894X(00)00423-6

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

We have described herein the syntheses of three novel series of aromatic ring containing pseudomycin side-chain analogues. Preliminary biological evaluations of these analogues clearly indicate that it is possible to synthesize rigid pseudomycin sidechain analogues without compromising in vitro antifungal activity. (C) 2000 Elsevier Science Ltd. All rights reserved.

引用

页码：2101 / 2105

页数：5

共 10 条

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