Bis-quinolinium cyclophanes:: 6,10-diaza-3(1,3),8(1,4)-dibenzena-1,5(1,4)-diquinolinacyclodecaphane (UCL 1684), the first nanomolar, non-peptidic blocker of the apamin-sensitive Ca2+-activated K+ channel

被引：72

作者：

Rosa, JC

Galanakis, D

Ganellin, CR

Dunn, PM

Jenkinson, DH

机构：

[1] Univ London Univ Coll, Christopher Ingold Labs, Dept Chem, London WC1H 0AJ, England

[2] UCL, Dept Chem, London WC1E 6BT, England

[3] UCL, Dept Pharmacol, London WC1E 6BT, England

[4] Univ Granada, Fac Farm, Dept Quim Organ, Granada 18071, Spain

[5] Aristotle Univ Thessaloniki, Sch Pharm, Dept Pharmaceut Chem, GR-54006 Thessaloniki, Greece

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1998年 / 41卷 / 01期

基金：

英国惠康基金;

关键词：

D O I：

10.1021/jm970571a

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：2 / 5

页数：4

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