In vivo and in vitro measurement of CYP2C19 activity

被引:12
作者
Wedlund, PJ [1 ]
Wilkinson, GR [1 ]
机构
[1] VANDERBILT UNIV,DEPT PHARMACOL,NASHVILLE,TN 37232
来源
CYTOCHROME P450, PT B | 1996年 / 272卷
关键词
D O I
10.1016/S0076-6879(96)72013-X
中图分类号
Q5 [生物化学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:105 / 114
页数:10
相关论文
共 21 条
  • [1] POLYMORPHIC HYDROXYLATION OF S-MEPHENYTOIN AND OMEPRAZOLE METABOLISM IN CAUCASIAN AND CHINESE SUBJECTS
    ANDERSSON, T
    REGARDH, CG
    LOU, YC
    ZHANG, Y
    DAHL, ML
    BERTILSSON, L
    [J]. PHARMACOGENETICS, 1992, 2 (01): : 25 - 31
  • [2] ARNS PA, 1990, PHARMACOLOGIST, V32, P140
  • [3] THE HYDROXYLATION OF OMEPRAZOLE CORRELATES WITH S-MEPHENYTOIN METABOLISM - A POPULATION STUDY
    BALIAN, JD
    SUKHOVA, N
    HARRIS, JW
    HEWETT, J
    PICKLE, L
    GOLDSTEIN, JA
    WOOSLEY, RL
    FLOCKHART, DA
    [J]. CLINICAL PHARMACOLOGY & THERAPEUTICS, 1995, 57 (06) : 662 - 669
  • [4] EXPRESSION OF A HUMAN-LIVER CYTOCHROME-P-450 PROTEIN WITH TOLBUTAMIDE HYDROXYLASE-ACTIVITY IN SACCHAROMYCES-CEREVISIAE
    BRIAN, WR
    SRIVASTAVA, PK
    UMBENHAUER, DR
    LLOYD, RS
    GUENGERICH, FP
    [J]. BIOCHEMISTRY, 1989, 28 (12) : 4993 - 4999
  • [5] Use of omeprazole as a probe drug for CYP2C19 phenotype in Swedish Caucasians: Comparison with S-mephenytoin hydroxylation phenotype and CYP2C19 genotype
    Chang, M
    Dahl, ML
    Tybring, G
    Gotharson, E
    Bertilsson, L
    [J]. PHARMACOGENETICS, 1995, 5 (06): : 358 - 363
  • [6] INTERPHENOTYPE DIFFERENCES IN DISPOSITION AND EFFECT ON GASTRIN-LEVELS OF OMEPRAZOLE - SUITABILITY OF OMEPRAZOLE AS A PROBE FOR CYP2C19
    CHANG, M
    TYBRING, G
    DAHL, ML
    GOTHARSON, E
    SAGAR, M
    SEENSALU, R
    BERTILSSON, L
    [J]. BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1995, 39 (05) : 511 - 518
  • [7] EVIDENCE THAT CYP2C19 IS THE MAJOR (S)-MEPHENYTOIN 4'-HYDROXYLASE IN HUMANS
    GOLDSTEIN, JA
    FALETTO, MB
    ROMKESSPARKS, M
    SULLIVAN, T
    KITAREEWAN, S
    RAUCY, JL
    LASKER, JM
    GHANAYEM, BI
    [J]. BIOCHEMISTRY, 1994, 33 (07) : 1743 - 1752
  • [8] GOLDSTEIN JA, 1996, METHODS ENZYMOL, V272, pCH23
  • [9] POLYMORPHIC METABOLISM OF MEPHENYTOIN IN MAN - PHARMACOKINETIC INTERACTION WITH A CO-REGULATED SUBSTRATE, MEPHOBARBITAL
    JACQZ, E
    HALL, SD
    BRANCH, RA
    WILKINSON, GR
    [J]. CLINICAL PHARMACOLOGY & THERAPEUTICS, 1986, 39 (06) : 646 - 653
  • [10] PHARMACOGENETICS OF MEPHENYTOIN - A NEW DRUG HYDROXYLATION POLYMORPHISM IN MAN
    KUPFER, A
    PREISIG, R
    [J]. EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1984, 26 (06) : 753 - 759