Discovery of (2S)-1-(4-amino-2,3,5-trimethylphenoxy)-3-{4-[4-(4-fluorobenzyl)phenyl]-1-piperazinyl}-2-propanol dimethanesulfonate (SUN N8075):: A dual Na+ and Ca2+ channel blocker with antioxidant activity

被引:22
作者
Annoura, H [1 ]
Nakanishi, K [1 ]
Toba, T [1 ]
Takemoto, N [1 ]
Imajo, S [1 ]
Miyajima, A [1 ]
Tamura-Horikawa, Y [1 ]
Tamura, S [1 ]
机构
[1] Suntory Biomed Res Ltd, Osaka 6188503, Japan
关键词
D O I
10.1021/jm000143w
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:3372 / 3376
页数:5
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