A very convenient dimethylamination of activated aromatic halides using N,N-dimethylformamide and ethanolamines

被引：42

作者：

Cho, YH ^{[1
]}

Park, JC ^{[1
]}

机构：

[1] HANHYO INST TECHNOL,PROC CHEM GRP,TAEJON 305390,SOUTH KOREA

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 48期

关键词：

D O I：

10.1016/S0040-4039(97)10255-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A very convenient dimethylamination of activated aromatic halides was achieved by using N,N-dimethylformamide(DMF) and ethanolamines. p-Nitrochlorobenzene, 2-halopyridines, 2-chloroquinoline and 2-chloropyrimidine gave the corresponding dimethylamino substituted products when treated with DMF and diethanolamine in 80 - 92% yield. (C) 1997 Elsevier Science Ltd.

引用

页码：8331 / 8334

页数：4

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