Hunting the emesis and efficacy targets of PDE4 inhibitors:: Identification of the photoaffinity probe 8-(3-azidophenyl)-6-[(4-iodo-1H-1-imidazolyl)methyl]quinoline (APIIMQ)

被引：28

作者：

Macdonald, D ^{[1
]}

Perrier, H ^{[1
]}

Liu, S ^{[1
]}

Laliberté, F ^{[1
]}

Rasori, R ^{[1
]}

Robichaud, A ^{[1
]}

Masson, P ^{[1
]}

Huang, Z ^{[1
]}

机构：

[1] Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 2000年 / 43卷 / 21期

关键词：

D O I：

10.1021/jm000065c

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：3820 / 3823

页数：4

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