Synthesis of substituted 2-mercaptobenzaldehydes and 2-substituted benzo[b]thiophenes

被引：32

作者：

Gallagher, T

Pardoe, DA

Porter, RA

机构：

[1] Univ Bristol, Sch Chem, Bristol BS8 1TS, Avon, England

[2] SB Pharmaceut, Discovery Res, Harlow CM19 5AW, Essex, England

来源：

TETRAHEDRON LETTERS | 2000年 / 41卷 / 28期

关键词：

D O I：

10.1016/S0040-4039(00)00870-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Simple and rapid single-pot preparations of substituted 2-mercaptobenzaldehydes 5 and 2-substituted benzo[b]thiophenes 3 based on ortho-lithiation methodology are described. (C) 2000 Elsevier Science Ltd. All rights reserved.

引用

页码：5415 / 5418

页数：4

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