Direct synthesis of 2-oxazolines from carboxylic acids using 2-chloro-4,6-dimethoxy-1,3,5-triazine under mild conditions

被引：63

作者：

Bandgar, BP ^{[1
]}

Pandit, SS ^{[1
]}

机构：

[1] Swami Ramanand Teerth Marathwada Univ, Sch Chem Sci, Organ Chem Res Lab, Vishnupuri 431606, Nanded, India

来源：

TETRAHEDRON LETTERS | 2003年 / 44卷 / 11期

关键词：

D O I：

10.1016/S0040-4039(03)00251-X

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

2-Acyloxy-4,6-dimethoxy-1,3,5-triazines obtained from carboxylic acids and 2-chloro-4,6-dimethoxy-1,3,5-triazine were subsequently treated with 2-amino-2-methyl-1-propanol to afford the corresponding 2-oxazolines in excellent yield at room temperature. (C) 2003 Published by Elsevier Science Ltd.

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页码：2331 / 2333

页数：3

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