Syntheses of 7-carboxyindolylglycines utilising glycine cation equivalents

被引:14
作者
Clark, BP [1 ]
Harris, JR [1 ]
机构
[1] ELI LILLY & CO,LILLY RES CTR LTD,WINDLESHAM GU20 6PH,SURREY,ENGLAND
关键词
D O I
10.1080/00397919708005046
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
The synthesis of two 7-carboxyindolylglycines is described as putative metabotropic glutamate receptor (mGluR) antagonists, employing glycine cation equivalents in the key steps.
引用
收藏
页码:4223 / 4234
页数:12
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