The dopamine D4 receptor:: a controversial therapeutic target

被引:33
作者
Hrib, NJ [1 ]
机构
[1] Aventis Pharmaceut, Dept Med Chem, Bridgewater, NJ 08807 USA
关键词
D O I
10.1358/dof.2000.025.06.858686
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:587 / 611
页数:25
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共 232 条
[71]   Binding of [3H]U-101958 to σ1 receptor-like sites in human cerebellum and neuroblastoma cells [J].
Helmeste, DM ;
Shioiri, T ;
Mitsuhashi, M ;
Tang, SW .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1999, 370 (02) :205-209
[72]   The naphtosultam derivative RP 62203 (fananserin) has high affinity for the dopamine D-4 receptor [J].
Heuillet, E ;
Petitet, F ;
Mignani, S ;
Malleron, JL ;
Lavayre, J ;
Neliat, G ;
Doble, A ;
Blanchard, JC .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1996, 314 (1-2) :229-233
[73]   YM-50001: A novel, potent and selective dopamine D4 receptor antagonist [J].
Hidaka, K ;
Tada, S ;
Matsumoto, M ;
Ohmori, J ;
Maeno, K ;
Yamaguchi, T .
NEUROREPORT, 1996, 7 (15-17) :2543-2546
[74]   Polymorphisms of dopamine receptor and transporter genes and Parkinson's disease [J].
Higuchi, S ;
Muramatsu, T ;
Arai, H ;
Hayashida, M ;
Sasaki, H ;
Trojanowski, JQ .
JOURNAL OF NEURAL TRANSMISSION-PARKINSONS DISEASE AND DEMENTIA SECTION, 1995, 10 (2-3) :107-113
[75]   Twelve-nucleotide repeat polymorphism of D4 dopamine receptor gene in Chinese familial schizophrenic patients [J].
Hong, CJ ;
Chiu, HJ ;
Chang, YS ;
Sim, CB .
BIOLOGICAL PSYCHIATRY, 1998, 43 (06) :432-435
[76]   Dopamine D4 receptor antagonist reversal of subchronic phencyclidine induced object retrieval detour deficits in monkeys [J].
Jentsch, JD ;
Taylor, JR ;
Redmond, DE ;
Elsworth, JD ;
Youngren, KD ;
Roth, RH .
PSYCHOPHARMACOLOGY, 1999, 142 (01) :78-84
[77]   A search for association between schizophrenia and dopamine-related alleles [J].
Jonsson, E ;
Brene, S ;
Geijer, T ;
Terenius, L ;
Tylec, A ;
Persson, ML ;
Sedvall, G .
EUROPEAN ARCHIVES OF PSYCHIATRY AND CLINICAL NEUROSCIENCE, 1996, 246 (06) :297-304
[78]  
Jonsson EG, 1997, AM J PSYCHIAT, V154, P697
[79]   Lack of association between dopamine D4 receptor gene and personality traits [J].
Jönsson, EG ;
Nöthen, MM ;
Gustavsson, JP ;
Neidt, H ;
Forslund, K ;
Mattila-Evenden, M ;
Rylander, G ;
Propping, P ;
Åsberg, M .
PSYCHOLOGICAL MEDICINE, 1998, 28 (04) :985-989
[80]   Drug therapy - Schizophrenia [J].
Kane, JM .
NEW ENGLAND JOURNAL OF MEDICINE, 1996, 334 (01) :34-41