Identification of a chemical tool for the orphan nuclear receptor FXR

被引：473

作者：

Maloney, PR

Parks, DJ

Haffner, CD

Fivush, AM

Chandra, G

Plunket, KD

Creech, KL

Moore, LB

Wilson, JG

Lewis, MC

Jones, SA

Willson, TM

机构：

[1] Glaxo Wellcome Res & Dev Ltd, Dept Med Chem, Res Triangle Pk, NC 27709 USA

[2] Glaxo Wellcome Res & Dev Ltd, Dept Mol Biochem, Res Triangle Pk, NC 27709 USA

[3] Glaxo Wellcome Res & Dev Ltd, Dept Mol Endocrinol, Res Triangle Pk, NC 27709 USA

[4] Glaxo Wellcome Res & Dev Ltd, Dept Metab Dis, Res Triangle Pk, NC 27709 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 2000年 / 43卷 / 16期

关键词：

D O I：

10.1021/jm0002127

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：2971 / 2974

页数：4

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