A new efficient synthesis of 3-(hydroxymethyl)-4H-chromen-4-ones

被引：13

作者：

Bolós, J ^{[1
]}

Loscertales, T ^{[1
]}

Nieto, J ^{[1
]}

Sacristán, A ^{[1
]}

Ortiz, JA ^{[1
]}

机构：

[1] Ctr Invest Grp Ferrer, Dept Med Chem, Barcelona 08028, Spain

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2000年 / 37卷 / 05期

关键词：

D O I：

10.1002/jhet.5570370529

中图分类号：

O62 [有机化学];

学科分类号：

070303 [有机化学]; 081704 [应用化学];

摘要：

An efficient and versatile synthesis of variously substituted 3-(hydroxymethyl)-4H-chromen-4-ones is reported. The compounds are prepared by hydroxymethylation of the precursor 2-hydroxy-4-chromanones followed by acid dehydration.

引用

页码：1203 / 1208

页数：6

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