Efficient nucleophilic substitution reaction of aryl halides with amino acids under focused microwave irradiation

被引：31

作者：

Cherng, YJ ^{[1
]}

机构：

[1] Chung Tai Inst Hlth Sci & Technol, Dept Med Technol, Taichung 40605, Taiwan

来源：

TETRAHEDRON | 2000年 / 56卷 / 42期

关键词：

microwave irradiation; nucleophilic aromatic substitution;

D O I：

10.1016/S0040-4020(00)00739-0

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The nucleophilic substitution reaction of 2,4-dinitrofluorobenzene with amino acids was complete, under microwave iradiation, within 40 s with yields up to 93%, which are far superior to those obtained under conventional heating. (C) 2000 Elsevier Science Ltd. All rights reserved.

引用

页码：8287 / 8289

页数：3

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