Copper-mediated cross-coupling reactions of N-unsubstituted sulfoximines and aryl halides

被引：102

作者：

Cho, GY ^{[1
]}

Rémy, P ^{[1
]}

Jansson, J ^{[1
]}

Moessner, C ^{[1
]}

Bolm, C ^{[1
]}

机构：

[1] Univ Aachen, Rhein Westfal TH Aachen, Inst Organ Chem, D-52056 Aachen, Germany

来源：

ORGANIC LETTERS | 2004年 / 6卷 / 19期

关键词：

D O I：

10.1021/ol048806h

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Copper-mediated cross-coupling reactions of sulfoximines with aryl iodides and aryl bromides provide N-arylated sulfoximines in high yields. The method is complementary to the known palladium-catalyzed N-arylation and allows the preparation of N-arylated sulfoximines, which have previously been inaccessible.

引用

页码：3293 / 3296

页数：4

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