Aminovinyl ketones and aminovinyl esters as C-C-N building blocks for the synthesis of 1H-pyrrolo[3,2-e]1,2,4-triazines

被引：25

作者：

Charushin, VN ^{[1
]}

Mochulskaya, NN

Andreiko, AA

Filyakova, VI

Kodess, MI

Chupakhin, ON

机构：

[1] Russian Acad Sci, Ural Branch, Inst Organ Synth, Ekaterinburg 620219, Russia

[2] Urals State Tech Univ, Dept Organ Chem, Ekaterinburg 620002, Russia

来源：

TETRAHEDRON LETTERS | 2003年 / 44卷 / 11期

基金：

俄罗斯基础研究基金会;

关键词：

1,2,4-triazines; tandem di-addition reactions; aminovinyl ketones; aminovinyl esters;

D O I：

10.1016/S0040-4039(03)00060-1

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

5,6-Unsubstituted-3-aryl-1,2,4-triazines were found to react with aminovinyl ketones and aminovinyl esters in acetic anhydride to form derivatives of 3a,4,7,7a-tetrahydro-1H-pyrrolo[3,2-e]1,2,4-triazines in good yields. (C) 2003 Elsevier Science Ltd. All rights reserved.

引用

页码：2421 / 2424

页数：4

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