Direct Pd-catalyzed arylation of 1,2,3-triazoles

被引：228

作者：

Chuprakov, Stepan ^{[1
]}

Chernyak, Natalia ^{[1
]}

Dudnik, Alexander S. ^{[1
]}

Gevorgyan, Vladimir ^{[1
]}

机构：

[1] Univ Illinois, Dept Chem, Chicago, IL 60607 USA

来源：

ORGANIC LETTERS | 2007年 / 9卷 / 12期

关键词：

D O I：

10.1021/ol070697u

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A highly efficient method for the synthesis of multisubstituted 1,2,3-triazoles via a direct Pd-catalyzed C-5 arylation has been developed.

引用

页码：2333 / 2336

页数：4

共 37 条

[1] ABBE G, 1969, IND CHIM BELG, V34, P519
[2] Aryl-aryl bond formation by transition-metal-catalyzed direct arylation
Alberico, Dino
Scott, Mark E.
Lautens, Mark
[J]. CHEMICAL REVIEWS, 2007, 107 (01) : 174 - 238
[3] 1,2,3-TRIAZOLE-[2',5'-BIS-O-(TERT-BUTYLDIMETHYLSILYL)-BETA-D-RIBOFURANOSYL]-3'-SPIRO-5''-(4''-AMINO-1'',2''-OXATHIOL 2'',2''-DIOXIDE) (TSAO) ANALOGS - SYNTHESIS AND ANTI-HIV-1 ACTIVITY
ALVAREZ, R
VELAZQUEZ, S
SANFELIX, A
AQUARO, S
DECLERCQ, E
PERNO, CF
KARLSSON, A
BALZARINI, J
CAMARASA, MJ
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1994, 37 (24) : 4185 - 4194
[4] Freeze-frame inhibitor captures acetylcholinesterase in a unique conformation
Bourne, Y
Kolb, HC
Radic, Z
Sharpless, KB
Taylor, P
Marchot, P
[J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2004, 101 (06) : 1449 - 1454
[5] An efficient access to 4-alkylidene-5,6-dihydro-4H-pyrrolo[1,2-c][1,2,3]triazoles
Chen, Wan-li
Su, Chen-liang
Huang, Xian
[J]. SYNLETT, 2006, (09) : 1446 - 1448
[6] Palladium-catalyzed arylation of electron-rich heterocycles with aryl chlorides
Chiong, Hendrich A.
Daugulis, Olafs
[J]. ORGANIC LETTERS, 2007, 9 (08) : 1449 - 1451
[7] Cross-coupling reaction of iodo-1,2,3-triazoles catalyzed by palladium
Deng, J
Wu, YM
Chen, QY
[J]. SYNTHESIS-STUTTGART, 2005, (16): : 2730 - 2738
[8] Fan W. Q., 1996, COMPREHENSIVE HETERO, V4, P1, DOI DOI 10.1016/B978-008096518-5.00079-4
[9] Felding J, 1998, SYNTHESIS-STUTTGART, P1181
[10] Reactivity and regioselectivity in the Heck reaction: Hammett study of 4-substituted styrenes
Fristrup, P
Le Quement, S
Tanner, D
Norrby, PO
[J]. ORGANOMETALLICS, 2004, 23 (26) : 6160 - 6165

← 1 2 3 4 →