Solid-phase synthesis of C-terminal peptide aldehydes from amino acetals anchored to a backbone amide linker (BAL) handle

被引：32

作者：

Guillaumie, F

Kappel, JC

Kelly, NM

Barany, G ^{[1
]}

Jensen, KJ

机构：

[1] Tech Univ Denmark, Dept Organ Chem, DK-2800 Lyngby, Denmark

[2] Univ Minnesota, Dept Chem, Minneapolis, MN 55455 USA

来源：

TETRAHEDRON LETTERS | 2000年 / 41卷 / 32期

基金：

美国国家卫生研究院;

关键词：

peptide aldehydes; solid-phase synthesis; BAL; amino acetals;

D O I：

10.1016/S0040-4039(00)00950-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：6131 / 6135

页数：5

共 15 条

[1] Ede NJ, 2000, J PEPT SCI, V6, P11, DOI 10.1002/(SICI)1099-1387(200001)6:1<11::AID-PSC229>3.0.CO
[2] 2-#
[3] FEHRENTZ JA, 1983, SYNTHESIS-STUTTGART, P676
[4] IMPROVED SOLID-PHASE SYNTHESIS OF C-TERMINAL PEPTIDE ALDEHYDES
FEHRENTZ, JA
PARIS, M
HEITZ, A
VELEK, J
LIU, CF
WINTERNITZ, F
MARTINEZ, J
[J]. TETRAHEDRON LETTERS, 1995, 36 (43) : 7871 - 7874
[5] Solid phase synthesis of C-terminal peptide aldehydes
Fehrentz, JA
Paris, M
Heitz, A
Velek, J
Winternitz, F
Martinez, J
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1997, 62 (20) : 6792 - 6796
[6] N-QUATERNARY COMPOUNDS .39. CIRCULAR-DICHROISM OF ALPHA-TRIMETHYLAMMONIO ALDEHYDES
GACEK, M
UNDHEIM, K
[J]. TETRAHEDRON, 1974, 30 (23-2) : 4233 - 4237
[7] Backbone Amide Linker (BAL) strategy for solid-phase synthesis of C-terminal-modified and cyclic peptides
Jensen, KJ
Alsina, J
Songster, MF
Vágner, J
Albericio, F
Barany, G
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1998, 120 (22) : 5441 - 5452
[8] NEW LEUPEPTIN ANALOGS - SYNTHESIS AND INHIBITION DATA
MCCONNELL, RM
BARNES, GE
HOYNG, CF
GUNN, JM
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1990, 33 (01) : 86 - 93
[9] AUTOMATED SYNTHESIS OF PEPTIDE C-TERMINAL ALDEHYDES
MURPHY, AM
DAGNINO, R
VALLAR, PL
TRIPPE, AJ
SHERMAN, SL
LUMPKIN, RH
TAMURA, SY
WEBB, TR
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1992, 114 (08) : 3156 - 3157
[10] Use of ozonolysis in the synthesis of C-terminal peptide aldehydes on solid support
Pothion, C
Paris, M
Heitz, A
Rocheblave, L
Rouch, F
Fehrentz, JA
Martinez, J
[J]. TETRAHEDRON LETTERS, 1997, 38 (44) : 7749 - 7752

← 1 2 →