Alkynylisothiazoles

被引：6

作者：

Zlotin, SG ^{[1
]}

Kislitsin, PG ^{[1
]}

Luk'yanov, OA ^{[1
]}

机构：

[1] Russian Acad Sci, ND Zelinskii Organ Chem Inst, Moscow 117913, Russia

来源：

RUSSIAN CHEMICAL BULLETIN | 1998年 / 47卷 / 03期

关键词：

haloisothiazoles; cross-coupling; palladium; acetylenes;

D O I：

10.1007/BF02495667

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A new synthesis of mono-and dialkynylisothiazoles by cross-coupling of bromine-and iodine-containing isothiazoles with terminal acetylene moieties in the PdCl2(PPh3)(2)-CuI-NEt3 catalytic system has been developed.

引用

页码：519 / 523

页数：5

共 30 条

[1] FACILE PALLADIUM-CATALYZED FUNCTIONALIZATION OF 1,2-ISOTHIAZOLINE-3-ONES [J].

BELL, AS ;

FISHWICK, CWG ;

REED, JE .

TETRAHEDRON LETTERS, 1994, 35 (35) :6551-6554

[2]

BLEICHER L, 1995, SYNLETT, P1115

[3]

Bohlmann F., 1973, NATURALLY OCCURING A

[4]

BREDAS JL, 1990, NATO ASI SER, V182

[5] (R)-(+)-N-[3-[5-[(4-FLUOROPHENYL)METHYL]-2-THIENYL]-1-METHYL-2-PROPYNYL]-N-HYDROXYUREA (ABT-761), A 2ND-GENERATION 5-LIPOXYGENASE INHIBITOR [J].

BROOKS, CDW ;

STEWART, AO ;

BASHA, A ;

BHATIA, P ;

RATAJCZYK, JD ;

MARTIN, JG ;

CRAIG, RA ;

KOLASA, T ;

BOUSKA, JB ;

LANNI, C ;

HARRIS, RR ;

MALO, PE ;

CARTER, GW ;

BELL, RL .

JOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (24) :4768-4775

[6]

BUMAGIN NA, 1982, DOKL AKAD NAUK SSSR+, V265, P1138

[7]

CHANDRARATNA RA, 1994, 13 INT S MED CHEM PA

[8] HEXAETHYNYLBENZENE [J].

DIERCKS, R ;

ARMSTRONG, JC ;

BOESE, R ;

VOLLHARDT, KPC .

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH, 1986, 25 (03) :268-269

[9] SYNTHESIS OF UNSYMMETRICAL 3,6-DISUBSTITUTED PYRIDAZINES - A PALLADIUM-CATALYZED APPROACH FROM 3-IODOPYRIDAZINES [J].

DRAPER, TL ;

BAILEY, TR .

JOURNAL OF ORGANIC CHEMISTRY, 1995, 60 (03) :748-750

[10]

Gopel W., 1992, NANOSTRUCTURES BASED

← 1 2 3 →