Synthesis of two new heteroaromatic β-carboline-fused pentacycles.: Observation of a new intercalating agent

被引：45

作者：

Csányi, D

Hajós, G

Riedl, Z

Timári, G

Bajor, Z

Cochard, F

Sapi, J

Laronze, JY

机构：

[1] Hungarian Acad Sci, Chem Res Ctr, Inst Chem, H-1525 Budapest, Hungary

[2] Univ Reims, Fac Pharm, CNRS,IFR Biomol 53, UPRESA Isolement Struct Transformat & Synth Prod, F-51096 Reims, France

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 2000年 / 10卷 / 15期

关键词：

D O I：

10.1016/S0960-894X(00)00339-5

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

Five-step synthetic routes of two new polyfused heterocycles: indazolo[3,2-a]-beta-carboline (3) and benzo[4',5'][1,2,3]triazino[6,1-a]-beta-carbolinium salt (10) applying Pd(0)-catalyzed cross-coupling reaction have been elaborated. (C) 2000 Elsevier Science Ltd. All rights reserved.

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页码：1767 / 1769

页数：3

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