A base labile handle for solid phase organic chemistry

被引：22

作者：

García-Echeverría, C ^{[1
]}

机构：

[1] Novartis Pharma Inc, Oncol Res, CH-4002 Basel, Switzerland

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 52期

关键词：

D O I：

10.1016/S0040-4039(97)10386-0

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Several arylsulfonamides have been synthesised on solid phase using a new bose labile handle. Cleavage from the solid support is accomplished by oxidation of the sulfide to the sulfone, followed by beta-elimination in base media. (C) 1997 Elsevier Science Ltd.

引用

页码：8933 / 8934

页数：2

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