Synthesis of 4-arylaminoquinazolines via 2-amino-N-arylbenzamidines

被引：35

作者：

Szczepankiewicz, W ^{[1
]}

Suwinski, J ^{[1
]}

机构：

[1] Silesian Tech Univ, Inst Organ Chem & Technol, PL-44100 Gliwice, Poland

来源：

TETRAHEDRON LETTERS | 1998年 / 39卷 / 13期

关键词：

D O I：

10.1016/S0040-4039(97)10864-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A new synthesis of twelve 4-arylaminoquinazolines from 2-amino-N-arylbenzamidines and formic acid is described. The entering amidines were obtained in the reaction of anthranilonitrile with 50% molar excess of aromatic amines and anhydrous aluminium chloride. (C) 1998 Elsevier Science Ltd. All rights reserved.

引用

页码：1785 / 1786

页数：2

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