Regulation of proteolytic activity by engineered tridentate metal binding loops

被引:20
作者
Halfon, S [1 ]
Craik, CS [1 ]
机构
[1] UNIV CALIF SAN FRANCISCO,DEPT PHARMACEUT CHEM,SAN FRANCISCO,CA 94143
关键词
D O I
10.1021/ja9533813
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
[No abstract available]
引用
收藏
页码:1227 / 1228
页数:2
相关论文
共 9 条
[1]  
BHOOLA KD, 1992, PHARMACOL REV, V44, P1
[2]   SILVER ION INHIBITION OF SERINE PROTEASES - CRYSTALLOGRAPHIC STUDY OF SILVER-TRYPSIN [J].
CHAMBERS, JL ;
CHRISTOPH, GG ;
KRIEGER, M ;
KAY, L ;
STROUD, RM .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1974, 59 (01) :70-74
[3]   RECENT ADVANCES IN THE EXPRESSION OF FOREIGN GENES IN PICHIA-PASTORIS [J].
CREGG, JM ;
VEDVICK, TS ;
RASCHKE, WC .
BIO-TECHNOLOGY, 1993, 11 (08) :905-910
[4]   ACITVATION INHIBITION AND PH-DEPENDENCE OF HYDROLYSIS OF ALPHA-N-BENZOYL-L-ARGININE ETHYL ESTER CATALYZED BY KALLIKREIN FROM PORCINE PANCREAS [J].
FIEDLER, F ;
WERLE, E .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1968, 7 (01) :27-&
[5]   RAT SUBMAXILLARY-GLAND SERINE PROTEASE, TONIN - STRUCTURE SOLUTION AND REFINEMENT AT 1.8 A RESOLUTION [J].
FUJINAGA, M ;
JAMES, MNG .
JOURNAL OF MOLECULAR BIOLOGY, 1987, 195 (02) :373-396
[6]   REGULATION OF SERINE PROTEASE ACTIVITY BY AN ENGINEERED METAL SWITCH [J].
HIGAKI, JN ;
HAYMORE, BL ;
CHEN, S ;
FLETTERICK, RJ ;
CRAIK, CS .
BIOCHEMISTRY, 1990, 29 (37) :8582-8586
[7]   THE 3-DIMENSIONAL STRUCTURE OF ASN102 MUTANT OF TRYPSIN - ROLE OF ASP102 IN SERINE PROTEASE CATALYSIS [J].
SPRANG, S ;
STANDING, T ;
FLETTERICK, RJ ;
STROUD, RM ;
FINERMOORE, J ;
XUONG, NH ;
HAMLIN, R ;
RUTTER, WJ ;
CRAIK, CS .
SCIENCE, 1987, 237 (4817) :905-909
[8]   HUMAN PROSTATE-SPECIFIC ANTIGEN - STRUCTURAL AND FUNCTIONAL SIMILARITY WITH SERINE PROTEASES [J].
WATT, KWK ;
LEE, PJ ;
MTIMKULU, T ;
CHAN, WP ;
LOOR, R .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (10) :3166-3170
[9]  
1971, STABILITY CONSTANT S, V1, P281