BCX-1812 (RWJ-270201): Discovery of a novel, highly potent, orally active, and selective influenza neuraminidase inhibitor through structure-based drug design

被引：346

作者：

Babu, YS

Chand, P

Bantia, S

Kotian, P

Dehghani, A

El-Kattan, Y

Lin, TH

Hutchison, TL

Elliott, AJ

Parker, CD

Ananth, SL

Horn, LL

Laver, GW

Montgomery, JA

机构：

[1] BioCryst Pharmaceut Inc, Birmingham, AL 35244 USA

[2] Australian Natl Univ, John Curtin Sch Med Res, Canberra, ACT 2601, Australia

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 2000年 / 43卷 / 19期

关键词：

D O I：

10.1021/jm0002679

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：3482 / 3486

页数：5

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