Novel orthogonal strategy toward solid-phase synthesis of 1,3,5-substituted triazines

被引：55

作者：

Bork, JT ^{[1
]}

Lee, JW ^{[1
]}

Khersonsky, SM ^{[1
]}

Moon, HS ^{[1
]}

Chang, YT ^{[1
]}

机构：

[1] NYU, Dept Chem, New York, NY 10003 USA

来源：

ORGANIC LETTERS | 2003年 / 5卷 / 02期

关键词：

D O I：

10.1021/ol027195v

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

To improve upon the previous orthogonal method for synthesis of a triazine library, an alternative strategy has been developed via oxidation-activation of the thioether to the sulfone. Through a comparison between these two methods, the sulfone strategy was demonstrated as an enhanced method in the generation of highly pure triazine library compounds.

引用

页码：117 / 120

页数：4

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