Application of AlMe3-mediated amidation reactions to solution phase peptide synthesis

被引：23

作者：

Martin, SF ^{[1
]}

Dwyer, MP ^{[1
]}

Lynch, CL ^{[1
]}

机构：

[1] Univ Texas, Dept Chem & Biochem, Austin, TX 78712 USA

来源：

TETRAHEDRON LETTERS | 1998年 / 39卷 / 12期

关键词：

D O I：

10.1016/S0040-4039(98)00071-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A practical modification of the Weinreb amidation protocol employing amino acids as the amine reaction partner has been developed that allows for the facile synthesis of oligopeptides in solution. (C) 1998 Elsevier Science Ltd. All rights reserved.

引用

页码：1517 / 1520

页数：4

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