Discovery of chiral N,N-disubstituted trifluoro-3-amino-2-propanols as potent inhibitors of cholesteryl ester transfer protein

被引：29

作者：

Durley, RC

Grapperhaus, ML

Massa, MA

Mischke, DA

Parnas, BL

Fobian, YM

Rath, NP

Honda, DD

Zeng, M

Connolly, DT

Heuvelman, DM

Witherbee, BJ

Glenn, KC

Krul, ES

Smith, ME

Sikorski, JA

机构：

[1] Pharmacia Discovery Res, St Louis, MO 63198 USA

[2] Univ Missouri, Dept Chem, St Louis, MO 63121 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 2000年 / 43卷 / 24期

关键词：

D O I：

10.1021/jm000337b

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：4575 / 4578

页数：4

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