Optically active arthropod repellents for use against disease vectors

被引：11

作者：

Klun, JA ^{[1
]}

Ma, D ^{[1
]}

Gupta, R ^{[1
]}

机构：

[1] ARS, Insect Chem Ecol Lab, USDA, Beltsville, MD 20705 USA

来源：

JOURNAL OF MEDICAL ENTOMOLOGY | 2000年 / 37卷 / 01期

关键词：

Anopheles stephensi; 1-[3-cyclohexen-1-ylcarbonyl] piperidine; 1-[3-cyclohexen-1-ylcarbonyl]-2-methylpiperidine; stereoisomers; repellents;

D O I：

10.1603/0022-2585-37.1.182

中图分类号：

Q96 [昆虫学];

学科分类号：

摘要：

Optically inactive 1-[3-cyclohexen-1-ylcarbonyl] piperidine and 1-[3-cyclohexen-1-ylcarbonyl]-2-methylpiperidine are repellents against blood-feeding arthropods. Pure stereoisomers of these compounds were synthesized. and characterized for use in bioassays. Initial laboratory tests with the malaria vector Anopheles stephensi Listen showed that this species was repelled differentially by the stereoisomers of 1-[3-cyclohexen-1-ylcarbonyl]-2-methylpiperidine. Two stereoisomers were twice as repellent as the other stereoisomers. These results indicate that stereoisomerism influences repellent efficacy in this class of compounds.

引用

页码：182 / 186

页数：5

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