Perspectives on the amorphisation/milling relationship in pharmaceutical materials

被引：131

作者：

Descamps, M. ^{[1
]}

Willart, J. F. ^{[1
]}

机构：

[1] Univ Lille, CNRS, Unite Mat & Transformat, UMET, F-59000 Lille, France

来源：

ADVANCED DRUG DELIVERY REVIEWS | 2016年 / 100卷

关键词：

Pharmaceuticals; Milling; Amorphous; Polymorphism; Phase transitions; SOLID-STATE AMORPHIZATION; PROCESS-INDUCED DISORDER; AMORPHOUS STATE; POLYMORPHIC TRANSFORMATION; ENTHALPY RELAXATION; GLASS-TRANSITION; REAL-TIME; IN-SITU; ENVIRONMENTAL-TEMPERATURE; INDOMETHACIN POLYMORPHS;

D O I：

10.1016/j.addr.2016.01.011

中图分类号：

R9 [药学];

学科分类号：

100702 [药剂学];

摘要：

This paper presents an overview of recent advances in understanding the role of the amorphous state in the physical and chemical transformations of pharmaceutical materials induced by mechanical milling. The following points are addressed: (1) Is milling really able to amorphise crystals?, (2) Conditions for obtaining an amorphisation, (3) Milling of hydrates, (4) Producing amorphous state without changing the chemical nature, (5) Milling induced crystal to crystal transformations: mediation by an amorphous state, (6) Nature of the amorphous state obtained by milling, (7) Milling of amorphous compounds: accelerated aging or rejuvenation, (8) Specific recrystallisation behaviour, and (9) Toward a rationalisation and conceptual framework. (c) 2016 Elsevier B.V. All rights reserved.

引用

页码：51 / 66

页数：16

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