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Ligands for glutamate receptors:: Design and therapeutic prospects
被引:522
作者
:
Bräuner-Osborne, H
论文数:
0
引用数:
0
h-index:
0
机构:
Royal Danish Sch Pharm, Dept Med Chem, NeuroSci PharmaBiotec Res Ctr, DK-2100 Copenhagen, Denmark
Bräuner-Osborne, H
Egebjerg, J
论文数:
0
引用数:
0
h-index:
0
机构:
Royal Danish Sch Pharm, Dept Med Chem, NeuroSci PharmaBiotec Res Ctr, DK-2100 Copenhagen, Denmark
Egebjerg, J
Nielsen, EO
论文数:
0
引用数:
0
h-index:
0
机构:
Royal Danish Sch Pharm, Dept Med Chem, NeuroSci PharmaBiotec Res Ctr, DK-2100 Copenhagen, Denmark
Nielsen, EO
Madsen, U
论文数:
0
引用数:
0
h-index:
0
机构:
Royal Danish Sch Pharm, Dept Med Chem, NeuroSci PharmaBiotec Res Ctr, DK-2100 Copenhagen, Denmark
Madsen, U
Krogsgaard-Larsen, P
论文数:
0
引用数:
0
h-index:
0
机构:
Royal Danish Sch Pharm, Dept Med Chem, NeuroSci PharmaBiotec Res Ctr, DK-2100 Copenhagen, Denmark
Krogsgaard-Larsen, P
机构
:
[1]
Royal Danish Sch Pharm, Dept Med Chem, NeuroSci PharmaBiotec Res Ctr, DK-2100 Copenhagen, Denmark
[2]
Aarhus Univ, Dept Mol & Struct Biol, DK-8000 Aarhus, Denmark
[3]
NeuroSearch AS, Dept Neurochem, DK-2750 Ballerup, Denmark
来源
:
JOURNAL OF MEDICINAL CHEMISTRY
|
2000年
/ 43卷
/ 14期
关键词
:
D O I
:
10.1021/jm000007r
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
[No abstract available]
引用
收藏
页码:2609 / 2645
页数:37
相关论文
共 418 条
[1]
Anti-epileptogenic and anticonvulsant activity of L-2-amino-4-phosphonobutyrate, a presynaptic glutamate receptor agonist
AbdulGhani, AS
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON IMPERIAL COLL SCI TECHNOL & MED,DEPT BIOCHEM,LONDON SW7 2AZ,ENGLAND
AbdulGhani, AS
Attwell, PJE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON IMPERIAL COLL SCI TECHNOL & MED,DEPT BIOCHEM,LONDON SW7 2AZ,ENGLAND
Attwell, PJE
Kent, NS
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON IMPERIAL COLL SCI TECHNOL & MED,DEPT BIOCHEM,LONDON SW7 2AZ,ENGLAND
Kent, NS
Bradford, HF
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON IMPERIAL COLL SCI TECHNOL & MED,DEPT BIOCHEM,LONDON SW7 2AZ,ENGLAND
Bradford, HF
Croucher, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON IMPERIAL COLL SCI TECHNOL & MED,DEPT BIOCHEM,LONDON SW7 2AZ,ENGLAND
Croucher, MJ
Jane, DE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON IMPERIAL COLL SCI TECHNOL & MED,DEPT BIOCHEM,LONDON SW7 2AZ,ENGLAND
Jane, DE
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Synthesis and pharmacological characterization of aminocyclopentanetricarboxylic acids: New tools to discriminate between metabotropic glutamate receptor subtypes
Acher, FC
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0
引用数:
0
h-index:
0
机构:
UNIV PARIS 05, CHIM & BIOCHIM PHARMACOL & TOXICOL LAB, CNRS, URA 400, F-75270 PARIS 06, FRANCE
Acher, FC
Tellier, FJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV PARIS 05, CHIM & BIOCHIM PHARMACOL & TOXICOL LAB, CNRS, URA 400, F-75270 PARIS 06, FRANCE
Tellier, FJ
Azerad, R
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV PARIS 05, CHIM & BIOCHIM PHARMACOL & TOXICOL LAB, CNRS, URA 400, F-75270 PARIS 06, FRANCE
Azerad, R
Brabet, IN
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UNIV PARIS 05, CHIM & BIOCHIM PHARMACOL & TOXICOL LAB, CNRS, URA 400, F-75270 PARIS 06, FRANCE
Brabet, IN
Fagni, L
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0
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0
h-index:
0
机构:
UNIV PARIS 05, CHIM & BIOCHIM PHARMACOL & TOXICOL LAB, CNRS, URA 400, F-75270 PARIS 06, FRANCE
Fagni, L
Pin, JPR
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0
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0
h-index:
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UNIV PARIS 05, CHIM & BIOCHIM PHARMACOL & TOXICOL LAB, CNRS, URA 400, F-75270 PARIS 06, FRANCE
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Corticolimbic dopamine neurotransmission is temporally dissociated from the cognitive and locomotor effects of phencyclidine
Adams, B
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0
引用数:
0
h-index:
0
机构:
Yale Univ, Sch Med, Vet Adm Med Ctr, Dept Psychiat, W Haven, CT 06516 USA
Yale Univ, Sch Med, Vet Adm Med Ctr, Dept Psychiat, W Haven, CT 06516 USA
Adams, B
Moghaddam, B
论文数:
0
引用数:
0
h-index:
0
机构:
Yale Univ, Sch Med, Vet Adm Med Ctr, Dept Psychiat, W Haven, CT 06516 USA
Yale Univ, Sch Med, Vet Adm Med Ctr, Dept Psychiat, W Haven, CT 06516 USA
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[J].
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Adler, CH
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0
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0
h-index:
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机构:
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
Adler, CH
Stern, MB
论文数:
0
引用数:
0
h-index:
0
机构:
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
Stern, MB
Vernon, G
论文数:
0
引用数:
0
h-index:
0
机构:
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
Vernon, G
Hurtig, HI
论文数:
0
引用数:
0
h-index:
0
机构:
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
Hurtig, HI
[J].
JOURNAL OF NEUROLOGY,
1997,
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(S)-Homo-AMPA, a specific agonist at the mGlu(6) subtype of metabotropic glutamic acid receptors
Ahmadian, H
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Ahmadian, H
Nielsen, B
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Nielsen, B
Brauner-Osborne, H
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Brauner-Osborne, H
Johansen, TN
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Johansen, TN
Stensbol, TB
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Stensbol, TB
Slok, FA
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Slok, FA
Sekiyama, N
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Sekiyama, N
Nakanishi, S
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Nakanishi, S
KrogsgaardLarsen, P
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
KrogsgaardLarsen, P
Madsen, U
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Madsen, U
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
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SYNTHESIS AND ACTIVITY OF A POTENT N-METHYL-D-ASPARTIC ACID AGONIST, TRANS-1-AMINOCYCLOBUTANE-1,3-DICARBOXYLIC ACID, AND RELATED PHOSPHONIC AND CARBOXYLIC-ACIDS
ALLAN, RD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
ALLAN, RD
HANRAHAN, JR
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
HANRAHAN, JR
HAMBLEY, TW
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0
引用数:
0
h-index:
0
机构:
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
HAMBLEY, TW
JOHNSTON, GAR
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UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
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0
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UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
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共 418 条
[1]
Anti-epileptogenic and anticonvulsant activity of L-2-amino-4-phosphonobutyrate, a presynaptic glutamate receptor agonist
AbdulGhani, AS
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON IMPERIAL COLL SCI TECHNOL & MED,DEPT BIOCHEM,LONDON SW7 2AZ,ENGLAND
AbdulGhani, AS
Attwell, PJE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON IMPERIAL COLL SCI TECHNOL & MED,DEPT BIOCHEM,LONDON SW7 2AZ,ENGLAND
Attwell, PJE
Kent, NS
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON IMPERIAL COLL SCI TECHNOL & MED,DEPT BIOCHEM,LONDON SW7 2AZ,ENGLAND
Kent, NS
Bradford, HF
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON IMPERIAL COLL SCI TECHNOL & MED,DEPT BIOCHEM,LONDON SW7 2AZ,ENGLAND
Bradford, HF
Croucher, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON IMPERIAL COLL SCI TECHNOL & MED,DEPT BIOCHEM,LONDON SW7 2AZ,ENGLAND
Croucher, MJ
Jane, DE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON IMPERIAL COLL SCI TECHNOL & MED,DEPT BIOCHEM,LONDON SW7 2AZ,ENGLAND
Jane, DE
[J].
BRAIN RESEARCH,
1997,
755
(02)
: 202
-
212
[2]
ABE T, 1992, J BIOL CHEM, V267, P13361
[3]
Synthesis and pharmacological characterization of aminocyclopentanetricarboxylic acids: New tools to discriminate between metabotropic glutamate receptor subtypes
Acher, FC
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV PARIS 05, CHIM & BIOCHIM PHARMACOL & TOXICOL LAB, CNRS, URA 400, F-75270 PARIS 06, FRANCE
Acher, FC
Tellier, FJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV PARIS 05, CHIM & BIOCHIM PHARMACOL & TOXICOL LAB, CNRS, URA 400, F-75270 PARIS 06, FRANCE
Tellier, FJ
Azerad, R
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV PARIS 05, CHIM & BIOCHIM PHARMACOL & TOXICOL LAB, CNRS, URA 400, F-75270 PARIS 06, FRANCE
Azerad, R
Brabet, IN
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV PARIS 05, CHIM & BIOCHIM PHARMACOL & TOXICOL LAB, CNRS, URA 400, F-75270 PARIS 06, FRANCE
Brabet, IN
Fagni, L
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV PARIS 05, CHIM & BIOCHIM PHARMACOL & TOXICOL LAB, CNRS, URA 400, F-75270 PARIS 06, FRANCE
Fagni, L
Pin, JPR
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV PARIS 05, CHIM & BIOCHIM PHARMACOL & TOXICOL LAB, CNRS, URA 400, F-75270 PARIS 06, FRANCE
Pin, JPR
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1997,
40
(19)
: 3119
-
3129
[4]
Adam G, 1999, NEUROPHARMACOLOGY, V38, pA1
[5]
Adam G., 1999, NEUROPHARMACOLOGY, V10, pA1
[6]
Corticolimbic dopamine neurotransmission is temporally dissociated from the cognitive and locomotor effects of phencyclidine
Adams, B
论文数:
0
引用数:
0
h-index:
0
机构:
Yale Univ, Sch Med, Vet Adm Med Ctr, Dept Psychiat, W Haven, CT 06516 USA
Yale Univ, Sch Med, Vet Adm Med Ctr, Dept Psychiat, W Haven, CT 06516 USA
Adams, B
Moghaddam, B
论文数:
0
引用数:
0
h-index:
0
机构:
Yale Univ, Sch Med, Vet Adm Med Ctr, Dept Psychiat, W Haven, CT 06516 USA
Yale Univ, Sch Med, Vet Adm Med Ctr, Dept Psychiat, W Haven, CT 06516 USA
Moghaddam, B
[J].
JOURNAL OF NEUROSCIENCE,
1998,
18
(14)
: 5545
-
5554
[7]
Amantadine in advanced Parkinson's disease: Good use of an old drug
Adler, CH
论文数:
0
引用数:
0
h-index:
0
机构:
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
Adler, CH
Stern, MB
论文数:
0
引用数:
0
h-index:
0
机构:
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
Stern, MB
Vernon, G
论文数:
0
引用数:
0
h-index:
0
机构:
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
Vernon, G
Hurtig, HI
论文数:
0
引用数:
0
h-index:
0
机构:
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
GRAD HOSP PHILADELPHIA,DEPT NEUROL,PHILADELPHIA,PA 19146
Hurtig, HI
[J].
JOURNAL OF NEUROLOGY,
1997,
244
(05)
: 336
-
337
[8]
(S)-Homo-AMPA, a specific agonist at the mGlu(6) subtype of metabotropic glutamic acid receptors
Ahmadian, H
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Ahmadian, H
Nielsen, B
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Nielsen, B
Brauner-Osborne, H
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Brauner-Osborne, H
Johansen, TN
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Johansen, TN
Stensbol, TB
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Stensbol, TB
Slok, FA
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Slok, FA
Sekiyama, N
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Sekiyama, N
Nakanishi, S
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Nakanishi, S
KrogsgaardLarsen, P
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
KrogsgaardLarsen, P
Madsen, U
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT MED CHEM, PHARMABIOTEC RES CTR, DK-2100 COPENHAGEN, DENMARK
Madsen, U
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1997,
40
(22)
: 3700
-
3705
[9]
SYNTHESIS AND ACTIVITY OF A POTENT N-METHYL-D-ASPARTIC ACID AGONIST, TRANS-1-AMINOCYCLOBUTANE-1,3-DICARBOXYLIC ACID, AND RELATED PHOSPHONIC AND CARBOXYLIC-ACIDS
ALLAN, RD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
ALLAN, RD
HANRAHAN, JR
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
HANRAHAN, JR
HAMBLEY, TW
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
HAMBLEY, TW
JOHNSTON, GAR
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
JOHNSTON, GAR
MEWETT, KN
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
MEWETT, KN
MITROVIC, AD
论文数:
0
引用数:
0
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机构:
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
UNIV SYDNEY, SCH CHEM, SYDNEY, NSW 2006, AUSTRALIA
MITROVIC, AD
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1990,
33
(10)
: 2905
-
2915
[10]
AMSTRONG N, 1998, NATURE, V395, P913
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