ANTI-CONVULSANT ACTIVITY OF GABA UPTAKE INHIBITORS AND THEIR PRODRUGS FOLLOWING CENTRAL OR SYSTEMIC ADMINISTRATION

被引:91
作者
CROUCHER, MJ
MELDRUM, BS
KROGSGAARDLARSEN, P
机构
[1] KINGS COLL HOSP MED SCH,RAYNE INST,DEPT NEUROL,LONDON SE5 9NU,ENGLAND
[2] ROYAL DANISH SCH PHARM,DEPT CHEM BC,DK-2100 COPENHAGEN O,DENMARK
关键词
D O I
10.1016/0014-2999(83)90497-1
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:217 / 228
页数:12
相关论文
共 32 条
  • [1] INHIBITION OF NEURONAL GABA UPTAKE AND GLIAL BETA-ALANINE UPTAKE BY SYNTHETIC GABA ANALOGS
    BRECKENRIDGE, RJ
    NICHOLSON, SH
    NICOL, AJ
    SUCKLING, CJ
    LEIGH, B
    IVERSEN, L
    [J]. BIOCHEMICAL PHARMACOLOGY, 1981, 30 (22) : 3045 - 3049
  • [2] BREHM L, 1979, GABA NEUROTRANSMITTE, P246
  • [3] CURTIS DR, 1976, EXP BRAIN RES, V25, P413
  • [4] CURTIS DR, 1974, ERG PHYSIOL BIOL CH, V69, P97
  • [5] CURTIS DR, 1979, GABA NEUROTRANSMITTE, P17
  • [6] AUDIOGENIC SEIZURE IN GENETICALLY SUSCEPTIBLE MICE - RELATION OF HYPOTHERMIA TO ONSET + SUSCEPTIBILITY
    ESSMAN, WB
    SUDAK, FN
    [J]. EXPERIMENTAL NEUROLOGY, 1964, 9 (03) : 228 - &
  • [7] INFLUENCE OF INHIBITORS OF THE HIGH-AFFINITY GABA UPTAKE ON SEIZURE THRESHOLDS IN MICE
    FREY, HH
    POPP, C
    LOSCHER, W
    [J]. NEUROPHARMACOLOGY, 1979, 18 (07) : 581 - 590
  • [8] THE EFFECT OF WETTING ON SOUND-INDUCED CONVULSIONS IN MICE
    FULLER, JL
    RAPPAPORT, A
    [J]. JOURNAL OF COMPARATIVE AND PHYSIOLOGICAL PSYCHOLOGY, 1952, 45 (04): : 246 - 249
  • [9] DRUG-INDUCED ELEVATION OF GABA AFTER INTRA-CEREBRAL MICRO-INJECTION - SITE OF ANTICONVULSANT ACTION
    GALE, K
    IADAROLA, M
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1980, 68 (02) : 233 - 235
  • [10] SYNAPTIC PHARMACOLOGY OF BARBITURATES AND BENZODIAZEPINES
    HAEFELY, WE
    [J]. AGENTS AND ACTIONS, 1977, 7 (03): : 353 - 359