EFFECT OF SELECTIVE 5HT3 ANTAGONIST (GR-38032F) ON SMALL INTESTINAL TRANSIT AND RELEASE OF GASTROINTESTINAL PEPTIDES

被引:47
作者
TALLEY, NJ [1 ]
PHILLIPS, SF [1 ]
HADDAD, A [1 ]
MILLER, LJ [1 ]
TWOMEY, C [1 ]
ZINSMEISTER, AR [1 ]
CIOCIOLA, A [1 ]
机构
[1] MAYO CLIN & MAYO FDN, CTR CORE, DIV GASTROENTEROL & DIGEST DIS, GASTROENTEROL UNIT, ROCHESTER, MN 55905 USA
关键词
D O I
10.1007/BF01537102
中图分类号
R57 [消化系及腹部疾病];
学科分类号
摘要
引用
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页码:1511 / 1515
页数:5
相关论文
共 25 条
[1]   EFFECT OF ICS 205-930 (A SPECIFIC 5-HT3 RECEPTOR ANTAGONIST) ON GASTRIC-EMPTYING OF A SOLID MEAL IN NORMAL SUBJECTS [J].
AKKERMANS, LMA ;
VOS, A ;
HOEKSTRA, A ;
ROELOFS, JMM ;
HOROWITZ, M .
GUT, 1988, 29 (09) :1249-1252
[2]  
BOND JH, 1975, J LAB CLIN MED, V85, P546
[3]   PROPOSALS FOR THE CLASSIFICATION AND NOMENCLATURE OF FUNCTIONAL RECEPTORS FOR 5-HYDROXYTRYPTAMINE [J].
BRADLEY, PB ;
ENGEL, G ;
FENIUK, W ;
FOZARD, JR ;
HUMPHREY, PPA ;
MIDDLEMISS, DN ;
MYLECHARANE, EJ ;
RICHARDSON, BP ;
SAXENA, PR .
NEUROPHARMACOLOGY, 1986, 25 (06) :563-576
[4]  
Bratton AC, 1939, J BIOL CHEM, V128, P537
[5]  
BRITTAIN R T, 1987, British Journal of Pharmacology, V90, p87P
[6]  
CARRAWAY R, 1976, J BIOL CHEM, V251, P7035
[7]  
CHANCE RC, 1977, METHOD HORM RADIOIMM, P657
[8]   PREVENTION OF EMESIS IN PATIENTS RECEIVING CYTOTOXIC DRUGS BY GR38032F, A SELECTIVE 5-HT3 RECEPTOR ANTAGONIST [J].
CUNNINGHAM, D ;
POPLE, A ;
FORD, HT ;
HAWTHORN, J ;
GAZET, JC ;
CHALLONER, T ;
COOMBES, RC .
LANCET, 1987, 1 (8548) :1461-1463
[9]  
DRYBURGH JR, 1975, GASTROENTEROLOGY, V68, P1169
[10]   NEURONAL 5-HT RECEPTORS IN THE PERIPHERY [J].
FOZARD, JR .
NEUROPHARMACOLOGY, 1984, 23 :1473-1486