SYNTHESIS OF DINUCLEOSIDE AND DINUCLEOTIDE PHOSPHORODITHIOATES VIA A PHOSPHOTRIESTER APPROACH

被引：40

作者：

YAU, EK ^{[1
]}

MA, YX ^{[1
]}

CARUTHERS, MH ^{[1
]}

机构：

[1] UNIV COLORADO,DEPT CHEM & BIOCHEM,BOULDER,CO 80309

来源：

TETRAHEDRON LETTERS | 1990年 / 31卷 / 14期

关键词：

D O I：

10.1016/S0040-4039(00)88887-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

5′ -O-Dimethoxytrityl and S-protected thymidine-3′ -phosphorodithioate, 3′ -O-acetylthymidine or thymidine-3′ -O-[β-cyanoethyl-(S-2,4-dichlorobenzyl)]-phosphorodithioate, 1-methylimidazole, and 2,4,6-triisopropylbenzenesulfonylchloride react to give excellent yields of dinucleoside phosphorodithioates. © 1990.

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页码：1953 / 1956

页数：4

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