PIPECOLIC ACIDS .3. SYNTHESIS OF UNNATURAL 2R,5S-5-HYDROXYPIPECOLIC ACID VIA HOMOCHIRAL ACYLIMINIUM ION

被引：34

作者：

HERDEIS, C

ENGEL, W

机构：

[1] Institut fur Pharmazie and Lebensmittelchemie der Universität 8700 Würzburg, Am Hubland

来源：

TETRAHEDRON-ASYMMETRY | 1991年 / 2卷 / 10期

关键词：

D O I：

10.1016/S0957-4166(00)86132-7

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

Stereoselective functionalization of S-5-hydroxy-2-piperidone 1 via acyliminium ion was demonstrated to maintain the unnatural enantiomer of trans-5-hydroxypipecolic acid 6.

引用

页码：945 / 948

页数：4

共 20 条

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[3] BEYERMAN HC, 1959, ARECL TRAV CHIM PAYS, V78, P648
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WAIBEL, D
[J]. ARCHIV DER PHARMAZIE, 1991, 324 (05) : 269 - 274
[7] HERDEIS C, IN PRESS ARCH PHARM
[8] KROGSGAARDLARSE.P, IN PRESS J NEUROCHEM
[9] REGIOSELECTIVE SYNTHESIS OF BETA-KETOESTERS FROM LITHIUM ENOLATES AND METHYL CYANOFORMATE
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[J]. TETRAHEDRON LETTERS, 1983, 24 (48) : 5425 - 5428
[10] INTRODUCTION OF ALKYL-GROUPS AT THE ALPHA-POSITIONS OF PYRROLIDINES AND PIPERIDINES - SYNTHESIS OF (+/-)-CONIINE
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[J]. HETEROCYCLES, 1988, 27 (07) : 1685 - 1696

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