EFFECTS OF THE BINDING OF IMIPRAMINE TO ERYTHROCYTES AND PLASMA-PROTEINS ON ITS TRANSPORT THROUGH THE RAT BLOOD-BRAIN-BARRIER

被引:30
作者
RIANT, P
URIEN, S
ALBENGRES, E
RENOUARD, A
TILLEMENT, JP
机构
关键词
D O I
10.1111/j.1471-4159.1988.tb01055.x
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
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页码:421 / 425
页数:5
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共 18 条
[1]   BINDING OF CHLORPROMAZINE AND IMIPRAMINE TO RED-CELLS, ALBUMIN, LIPOPROTEINS AND OTHER BLOOD COMPONENTS [J].
BICKEL, MH .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1975, 27 (10) :733-738
[2]  
CORNFORD EM, 1985, MOL PHYSIOL, V7, P219
[3]   BLOOD-BRAIN BARRIER TRANSPORT OF CI-912 - SINGLE-PASSAGE EQUILIBRATION OF ERYTHROCYTE-BORNE DRUG [J].
CORNFORD, EM ;
LANDON, KP .
THERAPEUTIC DRUG MONITORING, 1985, 7 (03) :247-254
[4]   PERMEABILITY OF CAPILLARIES IN VARIOUS ORGANS AS DETERMINED BY USE OF INDICATOR DIFFUSION METHOD [J].
CRONE, C .
ACTA PHYSIOLOGICA SCANDINAVICA, 1963, 58 (04) :292-&
[5]   OVERVIEW OF DRUG-PROTEIN BINDING [J].
GILLETTE, JR .
ANNALS OF THE NEW YORK ACADEMY OF SCIENCES, 1973, 226 (NOV26) :6-17
[6]   MULTIPLE HUMAN-SERUM BINDING OF 2 THIENOPYRIDINIC DERIVATIVES, TICLOPIDINE AND PCR 2362, AND THEIR DISTRIBUTION BETWEEN HSA, ALPHA-1-ACID GLYCOPROTEIN AND LIPOPROTEINS [J].
GLASSON, S ;
ZINI, R ;
TILLEMENT, JP .
BIOCHEMICAL PHARMACOLOGY, 1982, 31 (05) :831-835
[7]   EFFECT OF ERYTHROCYTES AND PLASMA-PROTEIN BINDING ON THE TRANSPORT OF PROGABIDE AND SL 75102 THROUGH THE RAT BLOOD-BRAIN-BARRIER [J].
HAMBERGER, C ;
URIEN, S ;
ESSASSI, D ;
GRIMALDI, B ;
BARRE, J ;
TAICLET, A ;
THENOT, JP ;
TILLEMENT, JP .
BIOCHEMICAL PHARMACOLOGY, 1987, 36 (16) :2641-2645
[8]   BRAIN UPTAKE OF RADIOLABELED AMINO ACIDS, AMINES, AND HEXOSES AFTER ARTERIAL INJECTION [J].
OLDENDORF, WH .
AMERICAN JOURNAL OF PHYSIOLOGY, 1971, 221 (06) :1629-+
[9]   TRANSPORT OF PROTEIN-BOUND HORMONES INTO TISSUES INVIVO [J].
PARDRIDGE, WM .
ENDOCRINE REVIEWS, 1981, 2 (01) :103-123
[10]   TRANSPORT OF PROPRANOLOL AND LIDOCAINE THROUGH THE RAT BLOOD-BRAIN-BARRIER - PRIMARY ROLE OF GLOBULIN-BOUND DRUG [J].
PARDRIDGE, WM ;
SAKIYAMA, R ;
FIERER, G .
JOURNAL OF CLINICAL INVESTIGATION, 1983, 71 (04) :900-908