BREMAZOCINE CAUSES SYMPATHO-INHIBITION AND HYPOTENSION IN RABBITS BY ACTIVATING PERIPHERAL KAPPA-RECEPTORS

被引:25
作者
ENSINGER, H [1 ]
HEDLER, L [1 ]
SZABO, B [1 ]
STARKE, K [1 ]
机构
[1] UNIV FREIBURG,INST PHARMAKOL,HERMANN HERDER STR 5,D-7800 FREIBURG,FED REP GER
关键词
D O I
10.1097/00005344-198605000-00005
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:470 / 475
页数:6
相关论文
共 25 条
[1]   IDENTIFICATION OF BENZOMORPHAN-K OPIATE RECEPTORS IN CEREBRAL-ARTERIES WHICH SUBSERVE RELAXATION [J].
ALTURA, BT ;
ALTURA, BM ;
QUIRION, R .
BRITISH JOURNAL OF PHARMACOLOGY, 1984, 82 (02) :459-466
[2]  
DHASMANA KM, 1982, ARCH INT PHARMACOD T, V260, P115
[3]   ETHYLKETOCYCLAZOCINE DECREASES NORADRENALINE RELEASE AND BLOOD-PRESSURE IN THE RABBIT AT A PERIPHERAL OPIOID RECEPTOR [J].
ENSINGER, H ;
HEDLER, L ;
SCHURR, C ;
STARKE, K .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1984, 328 (01) :20-23
[4]   MEASUREMENT OF TOTAL AND ORGAN-SPECIFIC NOREPINEPHRINE KINETICS IN HUMANS [J].
ESLER, M ;
JENNINGS, G ;
KORNER, P ;
BLOMBERY, P ;
SACHARIAS, N ;
LEONARD, P .
AMERICAN JOURNAL OF PHYSIOLOGY, 1984, 247 (01) :E21-E28
[5]   REDUCTION BY PHENTOLAMINE OF THE HYPOTENSIVE EFFECT OF METHIONINE ENKEPHALIN IN ANESTHETIZED RABBITS [J].
EULIE, PJ ;
RHEE, HM .
BRITISH JOURNAL OF PHARMACOLOGY, 1984, 83 (03) :783-790
[6]   DIFFERENTIAL CARDIOVASCULAR EFFECTS OF MU-OPIATE, DELTA-OPIATE AND KAPA-OPIATE AGONISTS AT DISCRETE HYPOTHALAMIC SITES IN THE ANESTHETIZED RAT [J].
FEUERSTEIN, G ;
FADEN, AI .
LIFE SCIENCES, 1982, 31 (20-2) :2197-2200
[7]  
GADDIS RR, 1982, J PHARMACOL EXP THER, V223, P77
[8]   PROFILE OF ACTIVITY OF KAPPA-RECEPTOR AGONISTS IN THE RABBIT VAS-DEFERENS [J].
HAYES, A ;
KELLY, A .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 110 (03) :317-322
[9]   MU, BUT NOT KAPPA, OPIOID AGONISTS INDUCE CONTRACTIONS OF THE CANINE SMALL-INTESTINE EXVIVO [J].
HIRNING, LD ;
PORRECA, F ;
BURKS, TF .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 109 (01) :49-54
[10]   INHIBITION OF NEUROEFFECTOR TRANSMISSION IN THE RABBIT MESENTERIC-ARTERY BY [MET5]ENKEPHALIN [J].
ILLES, P ;
RAMME, D ;
STARKE, K .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 107 (03) :397-398